Fragment Linking and Optimization of Inhibitors of the Aspartic Protease Endothiapepsin: Fragment-Based Drug Design Facilitated by Dynamic Combinatorial Chemistry
Mondal, Milon ; Radeva, Nedyalka ; Fanlo-Virgós, Hugo ; Otto, Sijbren ; Klebe, Gerhard ; Hirsch, Anna K. H.
Angewandte Chemie (International ed.), 2016-08, Vol.55 (32), p.9422-9426 [Periódico revisado por pares]Germany: Blackwell Publishing Ltd
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