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Material Type: Artigo
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Pep19 Has a Positive Effect on Insulin Sensitivity and Ameliorates Both Hepatic and Adipose Tissue Phenotype of Diet-Induced Obese MiceSilvério, Renata ; Barth, Robson ; Heimann, Andrea S ; Reckziegel, Patrícia ; Dos Santos, Gustavo J ; Romero-Zerbo, Silvana Y ; Bermúdez-Silva, Francisco J ; Rafacho, Alex ; Ferro, Emer SInternational journal of molecular sciences, 2022-04, Vol.23 (8), p.4082 [Periódico revisado por pares]Switzerland: MDPI AGTexto completo disponível |
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Material Type: Artigo
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Design, Synthesis, and Characterization of the Macrocyclic Tetrapeptide cyclo[Pro-Sar-Phe‑d‑Phe]: A Mixed Opioid Receptor Agonist–Antagonist Following Oral AdministrationFerracane, Michael J ; Brice-Tutt, Ariana C ; Coleman, Jeremy S ; Simpson, Grant G ; Wilson, Lisa L ; Eans, Shainnel O ; Stacy, Heather M ; Murray, Thomas F ; McLaughlin, Jay P ; Aldrich, Jane VACS chemical neuroscience, 2020-05, Vol.11 (9), p.1324-1336 [Periódico revisado por pares]United States: American Chemical SocietyTexto completo disponível |
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Material Type: Artigo
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Bradykinin antagonists: present progress and future prospectsStewart, John M ; Gera, Lajos ; York, Eunice J ; Chan, Daniel C ; Bunn, PaulImmunopharmacology, 1999-09, Vol.43 (2-3), p.155-161 [Periódico revisado por pares]Amsterdam: Elsevier B.VTexto completo disponível |
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Material Type: Artigo
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Form and Function in Cyclic Peptide Natural Products: A Pharmacokinetic PerspectiveBockus, Andrew T. ; McEwen, Cayla M. ; Lokey, R. ScottCurrent topics in medicinal chemistry, 2013-05, Vol.13 (7), p.821-836 [Periódico revisado por pares]Bentham Science Publishers LtdTexto completo disponível |
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Material Type: Artigo
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Dipteran toxicity assays for determining the oral insecticidal activity of venoms and toxinsGuo, Shaodong ; Herzig, Volker ; King, Glenn F.Toxicon (Oxford), 2018-08, Vol.150, p.297-303 [Periódico revisado por pares]England: Elsevier LtdTexto completo disponível |
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Material Type: Artigo
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Rational identification of a novel soy-derived anxiolytic-like undecapeptide acting via gut-brain axis after oral administrationOta, Ami ; Yamamoto, Akane ; Kimura, Saeko ; Mori, Yukiha ; Mizushige, Takafumi ; Nagashima, Yoshiki ; Sato, Masaru ; Suzuki, Hideyuki ; Odagiri, Saori ; Yamada, Daisuke ; Sekiguchi, Masayuki ; Wada, Keiji ; Kanamoto, Ryuhei ; Ohinata, KousakuNeurochemistry international, 2017-05, Vol.105, p.51-57 [Periódico revisado por pares]England: Elsevier LtdTexto completo disponível |
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7 |
Material Type: Artigo
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Design, synthesis, and biological activity of novel factor Xa inhibitors: Improving metabolic stability by S1 and S4 ligand modificationKomoriya, Satoshi ; Kobayashi, Shozo ; Osanai, Ken ; Yoshino, Toshiharu ; Nagata, Tsutomu ; Haginoya, Noriyasu ; Nakamoto, Yumi ; Mochizuki, Akiyoshi ; Nagahara, Takayasu ; Suzuki, Makoto ; Shimada, Takashi ; Watanabe, Kengo ; Isobe, Yumiko ; Furugoori, TaketoshiBioorganic & medicinal chemistry, 2006-03, Vol.14 (5), p.1309-1330 [Periódico revisado por pares]Oxford: Elsevier LtdTexto completo disponível |
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Material Type: Artigo
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RDP58, a locally active TNF inhibitor, is effective in the dextran sulphate mouse model of chronic colitisMurthy, S ; Flanigan, A ; Coppola, D ; Buelow, RInflammation research, 2002-11, Vol.51 (11), p.522-531 [Periódico revisado por pares]Switzerland: Springer Nature B.VTexto completo disponível |
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9 |
Material Type: Artigo
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Discovery of 1-[1-(1-Methylcyclooctyl)-4-piperidinyl]-2-[(3R)-3-piperidinyl]-1H-benzimidazole: Integrated Drug-Design and Structure-Activity Relationships for Orally Potent, Metabolically Stable and Potential-Risk Reduced Novel Non-Peptide Nociceptin/Orphanin FQ Receptor Agonist as Antianxiety Drug [double dagger]Hayashi, Shigeo ; Hirao, Akiko ; Nakamura, Hiroshi ; Yamamura, Kenzo ; Mizuno, Kunihiko ; Yamashita, HiroyoChemical biology & drug design, 2009-10, Vol.74 (4), p.369-381 [Periódico revisado por pares]Oxford, UK: Oxford, UK : Blackwell Publishing LtdTexto completo disponível |
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10 |
Material Type: Artigo
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Effects of an orally active non‐peptide bradykinin B2 receptor antagonist, FR173657, on plasma exudation in rat carrageenin‐induced pleurisyMajima, Masataka ; Kawashima, Noriko ; Hiroshi, Ito ; Katori, MakotoBritish journal of pharmacology, 1997-06, Vol.121 (4), p.723-730 [Periódico revisado por pares]Oxford, UK: Blackwell Publishing LtdTexto completo disponível |