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1 |
Material Type: Artigo
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Synthesis of indazole motifs and their medicinal importance: An overviewGaikwad, Digambar D. ; Chapolikar, Archana D. ; Devkate, Chandrashekhar G. ; Warad, Khandu D. ; Tayade, Amit P. ; Pawar, Rajendra P. ; Domb, Abraham J.European journal of medicinal chemistry, 2015-01, Vol.90, p.707-731 [Periódico revisado por pares]France: Elsevier Masson SASTexto completo disponível |
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Material Type: Artigo
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Recent progress in biological activities of synthesized phenothiazinesPluta, Krystian ; Morak-Młodawska, Beata ; Jeleń, MałgorzataEuropean journal of medicinal chemistry, 2011-08, Vol.46 (8), p.3179-3189 [Periódico revisado por pares]Kidlington: Elsevier Masson SASTexto completo disponível |
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Material Type: Artigo
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D 4 dopamine receptor high-resolution structures enable the discovery of selective agonistsWang, Sheng ; Wacker, Daniel ; Levit, Anat ; Che, Tao ; Betz, Robin M ; McCorvy, John D ; Venkatakrishnan, A J ; Huang, Xi-Ping ; Dror, Ron O ; Shoichet, Brian K ; Roth, Bryan LScience (American Association for the Advancement of Science), 2017-10, Vol.358 (6361), p.381-386 [Periódico revisado por pares]United States: AAASTexto completo disponível |
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Material Type: Artigo
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Zebrafish behavioral profiling identifies multitarget antipsychotic-like compoundsBruni, Giancarlo ; Rennekamp, Andrew J ; Velenich, Andrea ; McCarroll, Matthew ; Gendelev, Leo ; Fertsch, Ethan ; Taylor, Jack ; Lakhani, Parth ; Lensen, Dennis ; Evron, Tama ; Lorello, Paul J ; Huang, Xi-Ping ; Kolczewski, Sabine ; Carey, Galen ; Caldarone, Barbara J ; Prinssen, Eric ; Roth, Bryan L ; Keiser, Michael J ; Peterson, Randall T ; Kokel, DavidNature chemical biology, 2016-07, Vol.12 (7), p.559-566 [Periódico revisado por pares]United States: Nature Publishing GroupTexto completo disponível |
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Material Type: Artigo
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Antipsychotic Potential and Safety Profile of TPGS-Based Mucoadhesive Aripiprazole Nanoemulsion: Development and Optimization for Nose-To-Brain DeliveryKumbhar, Santosh Ashok ; Kokare, Chandrakant R. ; Shrivastava, Birendra ; Gorain, Bapi ; Choudhury, HiraJournal of pharmaceutical sciences, 2021-04, Vol.110 (4), p.1761-1778 [Periódico revisado por pares]United States: Elsevier IncSem texto completo |
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Material Type: Artigo
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Multi-Target Approach for Drug Discovery against SchizophreniaKondej, Magda ; Stępnicki, Piotr ; Kaczor, Agnieszka AInternational journal of molecular sciences, 2018-10, Vol.19 (10), p.3105 [Periódico revisado por pares]Switzerland: MDPITexto completo disponível |
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Material Type: Artigo
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Non-invasive intranasal delivery of quetiapine fumarate loaded microemulsion for brain targeting: Formulation, physicochemical and pharmacokinetic considerationShah, Brijesh ; Khunt, Dignesh ; Misra, Manju ; Padh, HarishEuropean journal of pharmaceutical sciences, 2016-08, Vol.91, p.196-207 [Periódico revisado por pares]Netherlands: Elsevier B.VTexto completo disponível |
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Material Type: Artigo
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Bioequivalence prediction with small-scale biphasic dissolution and simultaneous dissolution-permeation apparatus—An aripiprazole case studyKádár, Szabina ; Kennedy, Andrew ; Lee, Samuel ; Ruiz, Rebeca ; Farkas, Attila ; Tőzsér, Petra ; Csicsák, Dóra ; Tóth, Gergő ; Sinkó, Bálint ; Borbás, EnikőEuropean journal of pharmaceutical sciences, 2024-07, Vol.198, p.106782-106782, Article 106782 [Periódico revisado por pares]Netherlands: Elsevier B.VTexto completo disponível |
9 |
Material Type: Artigo
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Azaphenothiazines – promising phenothiazine derivatives. An insight into nomenclature, synthesis, structure elucidation and biological propertiesPluta, Krystian ; Jeleń, Małgorzata ; Morak-Młodawska, Beata ; Zimecki, Michał ; Artym, Jolanta ; Kocięba, Maja ; Zaczyńska, EwaEuropean journal of medicinal chemistry, 2017-09, Vol.138, p.774-806 [Periódico revisado por pares]France: Elsevier Masson SASTexto completo disponível |
10 |
Material Type: Artigo
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Enhanced dissolution, permeation and oral bioavailability of aripiprazole mixed micelles: In vitro and in vivo evaluationPiazzini, Vieri ; Landucci, Elisa ; Urru, Matteo ; Chiarugi, Alberto ; Pellegrini-Giampietro, Domenico E. ; Bilia, Anna Rita ; Bergonzi, Maria CamillaInternational journal of pharmaceutics, 2020-06, Vol.583, p.119361, Article 119361 [Periódico revisado por pares]Netherlands: Elsevier B.VTexto completo disponível |