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Design, synthesis, structural optimization, SAR, in silico prediction of physicochemical properties and pharmacological evaluation of novel & potent thiazolo[4,5-d]pyrimidine corticotropin releasing factor (CRF) receptor antagonists
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Design, synthesis, structural optimization, SAR, in silico prediction of physicochemical properties and pharmacological evaluation of novel & potent thiazolo[4,5-d]pyrimidine corticotropin releasing factor (CRF) receptor antagonists

Islam, Md Rabiul ; Teleb, Mohamed ; Karageorgos, Vlasios ; Sakellaris, Stelios ; Papadopoulos, Minas ; Pirmettis, Ioannis ; Fronczek, Frank R. ; Liapakis, George ; Fahmy, Hesham

European journal of pharmaceutical sciences, 2022-02, Vol.169, p.106084-106084, Article 106084 [Periódico revisado por pares]

Netherlands: Elsevier B.V

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2
Crinecerfont in a First Clinical Application of a CRH Antagonist: Further Potential Uses Are Still an Open Chapter
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Crinecerfont in a First Clinical Application of a CRH Antagonist: Further Potential Uses Are Still an Open Chapter

Chrousos, George P

The journal of clinical endocrinology and metabolism, 2024-03, Vol.109 (4), p.e1365-e1366 [Periódico revisado por pares]

United States

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3
Activation of NOP receptor increases vulnerability to stress: role of glucocorticoids and CRF signaling
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Artigo
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Activation of NOP receptor increases vulnerability to stress: role of glucocorticoids and CRF signaling

Holanda, Victor A. D. ; de Almeida, Raissa N. ; de Oliveira, Matheus C ; da Silva Junior, Edilson D. ; Galvão-Coelho, Nicole L. ; Calo’, Girolamo ; Ruzza, Chiara ; Gavioli, Elaine C.

Psychopharmacology, 2024-05, Vol.241 (5), p.1001-1010 [Periódico revisado por pares]

Berlin/Heidelberg: Springer Berlin Heidelberg

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4
Amino acid systems in the interpeduncular nucleus are altered in a sex‐dependent manner during nicotine withdrawal
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Artigo
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Amino acid systems in the interpeduncular nucleus are altered in a sex‐dependent manner during nicotine withdrawal

Carcoba, Luis M. ; Uribe, Kevin P. ; Ortegon, Sebastian ; Mendez, Ian A. ; DeBiasi, Mariella ; O'Dell, Laura E.

Journal of neuroscience research, 2022-08, Vol.100 (8), p.1573-1584 [Periódico revisado por pares]

United States: Wiley Subscription Services, Inc

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5
The effects of alcohol on anxiety-like, depression-like, and social behavior immediately and a day after binge drinking
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Artigo
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The effects of alcohol on anxiety-like, depression-like, and social behavior immediately and a day after binge drinking

Simon, Balázs ; Thury, Attila Ágoston ; Török, László ; Földesi, Imre ; Csabafi, Krisztina ; Bagosi, Zsolt

Alcohol (Fayetteville, N.Y.), 2023-11, Vol.112, p.17-24 [Periódico revisado por pares]

United States: Elsevier Inc

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6
Corticotropin-releasing factor regulates caspase-3 and may protect developing zebrafish from stress-induced apoptosis
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Corticotropin-releasing factor regulates caspase-3 and may protect developing zebrafish from stress-induced apoptosis

Alderman, Sarah L. ; Leishman, Emily M. ; Fuzzen, Meghan L.M. ; Bernier, Nicholas J.

General and comparative endocrinology, 2018-09, Vol.265, p.207-213 [Periódico revisado por pares]

United States: Elsevier Inc

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7
Dopamine and Stress System Modulation of Sex Differences in Decision Making
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Dopamine and Stress System Modulation of Sex Differences in Decision Making

Georgiou, Polymnia ; Zanos, Panos ; Bhat, Shambhu ; Tracy, J Kathleen ; Merchenthaler, Istvan J ; McCarthy, Margaret M ; Gould, Todd D

Neuropsychopharmacology (New York, N.Y.), 2018-01, Vol.43 (2), p.313-324 [Periódico revisado por pares]

England: Nature Publishing Group

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8
Beyond depression and anxiety; a systematic review about the role of corticotropin-releasing hormone antagonists in diseases of the pelvic and abdominal organs
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Beyond depression and anxiety; a systematic review about the role of corticotropin-releasing hormone antagonists in diseases of the pelvic and abdominal organs

Pagán-Busigó, Joshua E ; López-Carrasquillo, Jonathan ; Appleyard, Caroline B ; Torres-Reverón, Annelyn Reichmann, Florian

PloS one, 2022-03, Vol.17 (3), p.e0264909-e0264909 [Periódico revisado por pares]

United States: Public Library of Science

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9
Drug addiction: the neurobiology of behaviour gone awry
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Drug addiction: the neurobiology of behaviour gone awry

Volkow, Nora D ; Li, Ting-Kai

Nature reviews. Neuroscience, 2004-12, Vol.5 (12), p.963-970 [Periódico revisado por pares]

London: Nature Publishing Group

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10
Sex‐linked roles of the CRF1 and the CRF2 receptor in social behavior
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Sex‐linked roles of the CRF1 and the CRF2 receptor in social behavior

Piccin, Alessandro ; Contarino, Angelo

Journal of neuroscience research, 2020-08, Vol.98 (8), p.1561-1574 [Periódico revisado por pares]

Hoboken: Wiley Subscription Services, Inc

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