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Material Type: Artículo
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Mechanisms of signalling and biased agonism in G protein-coupled receptorsWootten, Denise ; Christopoulos, Arthur ; Marti-Solano, Maria ; Babu, M Madan ; Sexton, Patrick MNature reviews. Molecular cell biology, 2018-10, Vol.19 (10), p.638-653 [Revista revisada por pares]England: Nature Publishing GroupTexto completo disponible |
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Material Type: Artículo
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Structure, function and pharmacology of human itch GPCRsCao, Can ; Kang, Hye Jin ; Singh, Isha ; Chen, He ; Zhang, Chengwei ; Ye, Wenlei ; Hayes, Byron W ; Liu, Jing ; Gumpper, Ryan H ; Bender, Brian J ; Slocum, Samuel T ; Krumm, Brian E ; Lansu, Katherine ; McCorvy, John D ; Kroeze, Wesley K ; English, Justin G ; DiBerto, Jeffrey F ; Olsen, Reid H J ; Huang, Xi-Ping ; Zhang, Shicheng ; Liu, Yongfeng ; Kim, Kuglae ; Karpiak, Joel ; Jan, Lily Y ; Abraham, Soman N ; Jin, Jian ; Shoichet, Brian K ; Fay, Jonathan F ; Roth, Bryan LNature (London), 2021-12, Vol.600 (7887), p.170-175 [Revista revisada por pares]England: Nature Publishing GroupTexto completo disponible |
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Material Type: Artículo
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Conformational Basis of G Protein-Coupled Receptor Signaling VersatilityWingler, Laura M. ; Lefkowitz, Robert J.Trends in cell biology, 2020-09, Vol.30 (9), p.736-747 [Revista revisada por pares]England: Elsevier LtdTexto completo disponible |
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Material Type: Artículo
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GPCRomics: An Approach to Discover GPCR Drug TargetsInsel, Paul A. ; Sriram, Krishna ; Gorr, Matthew W. ; Wiley, Shu Z. ; Michkov, Alexander ; Salmerón, Cristina ; Chinn, Amy M.Trends in pharmacological sciences (Regular ed.), 2019-06, Vol.40 (6), p.378-387 [Revista revisada por pares]England: Elsevier LtdTexto completo disponible |
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Material Type: Artículo
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Structural insights into G-protein-coupled receptor allosteryThal, David M ; Glukhova, Alisa ; Sexton, Patrick M ; Christopoulos, ArthurNature (London), 2018-07, Vol.559 (7712), p.45-53 [Revista revisada por pares]England: Nature Publishing GroupTexto completo disponible |
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Material Type: Artículo
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THE CONCISE GUIDE TO PHARMACOLOGY 2019/20: G protein‐coupled receptorsAlexander, Stephen PH ; Davenport, Anthony P ; Peters, John A ; Veale, Emma L ; Faccenda, Elena ; Harding, Simon D ; Pawson, Adam J ; Sharman, Joanna L ; Southan, Christopher ; Abbracchio, Maria P ; Alexander, Wayne ; Al-hosaini, Khaled ; Bäck, Magnus ; Beaulieu, Jean‐Martin ; Bernstein, Kenneth E. ; Birdsall, Nigel JM ; Blaho, Victoria ; Bousquet, Corinne ; Caló, Girolamo ; Ceruti, Stefania ; Chazot, Paul ; Chiang, Nan ; Chun, Jerold ; Cianciulli, Antonia ; Clapp, Lucie H ; Couture, Réjean ; Dent, Gordon ; Douglas, Steven D ; Dournaud, Pascal ; Eguchi, Satoru ; Filardo, Edward ; Fong, Tung M ; Fumagalli, Marta ; Gainetdinov, Raul R ; Gasparo, Marc de ; Goudet, Cyril ; Gregory, Karen J ; Hamann, Jörg ; Hauger, Richard L ; Heinemann, Akos ; Holliday, Nicholas D ; Horiuchi, Mastgugu ; Husain, Ahsan ; Inagami, Tadashi ; Jacobson, Kenneth A ; Jensen, Robert T ; Jockers, Ralf ; Jonnalagadda, Deepa ; Kemp, Jacqueline ; Kennedy, Charles ; Kihara, Yasuyuki ; Kukkonen, Jyrki P ; Leach, Katie ; Lecca, Davide ; Lee, John D ; Leeman, Susan E ; Leprince, Jérôme ; Lolait, Stephen J ; Lupp, Amelie ; Macrae, Robyn ; Mazella, Jean ; McArdle, Craig A ; Melmed, Shlomo ; Michel, Martin C ; Miller, Laurence ; Mitolo, Vincenzo ; Mouillac, Bernard ; Murphy, Philip M ; Nahon, Jean‐Louis ; Norel, Xavier ; Nyimanu, Duuamene ; O'Carroll, Anne‐Marie ; Panaro, Maria A ; Pertwee, Roger G ; Pin, Jean‐Philippe ; Prossnitz, Eric ; Rovati, G Enrico ; Ruzza, Chiara ; Sanger, Gareth ; Schöneberg, Torsten ; Schulte, Gunnar ; Serhan, Charles N ; Stoddart, Leigh A ; Sugimoto, Yukihiko ; Summers, Roger ; Tan, Valerie ; Thomas, Walter ; Tirupula, Kalyan ; Tulipano, Giovanni ; Unal, Hamiyet ; Unger, Thomas ; Vanderheyden, Patrick ; Vilardaga, Jean‐Pierre ; Walker, Christopher S ; Ward, Donald T ; Wester, Hans‐Jürgen ; Willars, Gary B ; Williams, Tom Lloyd ; Woodruff, Trent M ; Yao, ChengcanBritish journal of pharmacology, 2019-12, Vol.176 (S1), p.S21-S141 [Revista revisada por pares]England: Blackwell Publishing LtdTexto completo disponible |
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Material Type: Artículo
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Differential GLP-1R Binding and Activation by Peptide and Non-peptide AgonistsZhang, Xin ; Belousoff, Matthew J. ; Zhao, Peishen ; Kooistra, Albert J. ; Truong, Tin T. ; Ang, Sheng Yu ; Underwood, Christina Rye ; Egebjerg, Thomas ; Šenel, Petr ; Stewart, Gregory D. ; Liang, Yi-Lynn ; Glukhova, Alisa ; Venugopal, Hari ; Christopoulos, Arthur ; Furness, Sebastian G.B. ; Miller, Laurence J. ; Reedtz-Runge, Steffen ; Langmead, Christopher J. ; Gloriam, David E. ; Danev, Radostin ; Sexton, Patrick M. ; Wootten, DeniseMolecular cell, 2020-11, Vol.80 (3), p.485-500.e7 [Revista revisada por pares]United States: Elsevier IncTexto completo disponible |
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8 |
Material Type: Artículo
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DREADDs (Designer Receptors Exclusively Activated by Designer Drugs): Chemogenetic Tools with Therapeutic UtilityUrban, Daniel J ; Roth, Bryan LAnnual review of pharmacology and toxicology, 2015-01, Vol.55 (1), p.399-417 [Revista revisada por pares]United States: Annual ReviewsTexto completo disponible |
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Material Type: Artículo
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GPCR-G Protein-β-Arrestin Super-Complex Mediates Sustained G Protein SignalingThomsen, Alex R.B. ; Plouffe, Bianca ; Cahill, Thomas J. ; Shukla, Arun K. ; Tarrasch, Jeffrey T. ; Dosey, Annie M. ; Kahsai, Alem W. ; Strachan, Ryan T. ; Pani, Biswaranjan ; Mahoney, Jacob P. ; Huang, Liyin ; Breton, Billy ; Heydenreich, Franziska M. ; Sunahara, Roger K. ; Skiniotis, Georgios ; Bouvier, Michel ; Lefkowitz, Robert J.Cell, 2016-08, Vol.166 (4), p.907-919 [Revista revisada por pares]United States: Elsevier IncTexto completo disponible |
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10 |
Material Type: Artículo
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GPCRdb in 2018: adding GPCR structure models and ligandsPándy-Szekeres, Gáspár ; Munk, Christian ; Tsonkov, Tsonko M ; Mordalski, Stefan ; Harpsøe, Kasper ; Hauser, Alexander S ; Bojarski, Andrzej J ; Gloriam, David ENucleic acids research, 2018-01, Vol.46 (D1), p.D440-D446 [Revista revisada por pares]England: Oxford University PressTexto completo disponible |