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1
1-(2-METHOXYPHENYL)-4-ALKYLPIPERAZINES: EFFECT OF THE N-4 SUBSTITUENT ON THE AFFINITY AND SELECTIVITY FOR DOPAMINE D 4 RECEPTOR
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1-(2-METHOXYPHENYL)-4-ALKYLPIPERAZINES: EFFECT OF THE N-4 SUBSTITUENT ON THE AFFINITY AND SELECTIVITY FOR DOPAMINE D 4 RECEPTOR

Perrone, Roberto ; Berardi, Francesco ; Colabufo, Nicola A ; Leopoldo, Marcello ; Tortorella, Vincenzo

Bioorganic & medicinal chemistry letters, 1997-05, Vol.7 (10), p.1327-1330 [Periódico revisado por pares]

Elsevier Ltd

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2
1-(3-Cyanobenzylpiperidin-4-yl)-5-methyl-4-phenyl-1,3-dihydroimidazol-2-one:  A Selective High-Affinity Antagonist for the Human Dopamine D 4 Receptor with Excellent Selectivity over Ion Channels
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1-(3-Cyanobenzylpiperidin-4-yl)-5-methyl-4-phenyl-1,3-dihydroimidazol-2-one:  A Selective High-Affinity Antagonist for the Human Dopamine D 4 Receptor with Excellent Selectivity over Ion Channels

Carling, Robert W. ; Moore, Kevin W. ; Moyes, Christopher R. ; Jones, Elizabeth A. ; Bonner, Katrine ; Emms, Frances ; Marwood, Rosemary ; Patel, Shil ; Patel, Smita ; Fletcher, Alan E. ; Beer, Margaret ; Sohal, Bindi ; Pike, Andrew ; Leeson, Paul D.

Journal of medicinal chemistry, 1999-07, Vol.42 (14), p.2706-2715 [Periódico revisado por pares]

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3
1,2-Addition to trifluoromethylated β-enamino diketones: regioselective synthesis of trifluoromethyl-containing azomethine pyrazoles and isoxazoles
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1,2-Addition to trifluoromethylated β-enamino diketones: regioselective synthesis of trifluoromethyl-containing azomethine pyrazoles and isoxazoles

Pianoski, Karlos Eduardo ; Poletto, Julia ; Vieira da Silva, Michael Jackson ; Ascencio Camargo, Jeniffer Nascimento ; Jacomini, Andrey Petita ; Gonçalves, Davana Silva ; Back, Davi Fernando ; Moura, Sidnei ; Rosa, Fernanda Andreia

Organic & biomolecular chemistry, 2020-04, Vol.18 (13), p.2524-2537 [Periódico revisado por pares]

England: Royal Society of Chemistry

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4
1,2-Diastereoselective C-C Bond-Forming Reactions for the Synthesis of Chiral β-Branched α-Amino Acids
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1,2-Diastereoselective C-C Bond-Forming Reactions for the Synthesis of Chiral β-Branched α-Amino Acids

Spangenberg, Thomas ; Schoenfelder, Angèle ; Breit, Bernhard ; Mann, André

European Journal of Organic Chemistry, 2010-11, Vol.2010 (31), p.6005-6018 [Periódico revisado por pares]

Weinheim: WILEY-VCH Verlag

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5
1.2-kV Low-Barrier 4H-SiC JBS Diodes by Virtue of P-Implants Across Dead Field of Current Flow
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1.2-kV Low-Barrier 4H-SiC JBS Diodes by Virtue of P-Implants Across Dead Field of Current Flow

Zhang, Yuan-Lan ; Liu, Pan ; Lei, Guang-Yin ; Zhang, Qingchun J.

IEEE transactions on electron devices, 2023-08, Vol.70 (8), p.4293-4302 [Periódico revisado por pares]

IEEE

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6
1,2,3-Triazole-containing hybrids as potential anticancer agents: Current developments, action mechanisms and structure-activity relationships
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1,2,3-Triazole-containing hybrids as potential anticancer agents: Current developments, action mechanisms and structure-activity relationships

Xu, Zhi ; Zhao, Shi-Jia ; Liu, Yi

European journal of medicinal chemistry, 2019-12, Vol.183, p.111700-111700, Article 111700 [Periódico revisado por pares]

France: Elsevier Masson SAS

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7
1,2,3,4-Tetrahydroisoquinoline/2H-chromen-2-one conjugates as nanomolar P-glycoprotein inhibitors: Molecular determinants for affinity and selectivity over multidrug resistance associated protein 1
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1,2,3,4-Tetrahydroisoquinoline/2H-chromen-2-one conjugates as nanomolar P-glycoprotein inhibitors: Molecular determinants for affinity and selectivity over multidrug resistance associated protein 1

Rullo, Mariagrazia ; Niso, Mauro ; Pisani, Leonardo ; Carrieri, Antonio ; Colabufo, Nicola Antonio ; Cellamare, Saverio ; Altomare, Cosimo Damiano

European journal of medicinal chemistry, 2019-01, Vol.161, p.433-444 [Periódico revisado por pares]

France: Elsevier Masson SAS

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8
1,2,4-triazole-5-thione derivative for inhibiting carbon steel corrosion in 1M HCl: Synthesis, electrochemical, SEM/EDX, DFT, and MD investigations
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1,2,4-triazole-5-thione derivative for inhibiting carbon steel corrosion in 1M HCl: Synthesis, electrochemical, SEM/EDX, DFT, and MD investigations

Rehioui, Malak ; Lazrak, Fatima ; Lahmidi, Sanae ; Benmekki, Saad ; El-Yazeed, Wafaa S. Abo ; Anouar, El Hassane ; Erramli, Hamid ; Hajjaji, Najat

Journal of molecular structure, 2024-05, Vol.1303, p.137577, Article 137577 [Periódico revisado por pares]

Elsevier B.V

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9
[1,2,4]triazole derivatives as 5-HT1A serotonin receptor ligands
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[1,2,4]triazole derivatives as 5-HT1A serotonin receptor ligands

SARVA, Maria Concetta ; ROMEO, Giuseppe ; GUERRERA, Francesco ; SIRACUSA, Mariangela ; SALERNO, Loredana ; RUSSO, Filippo ; CAGNOTTO, Alfredo ; GOEGAN, Mara ; MENNINI, Tiziana

Bioorganic & medicinal chemistry, 2002-02, Vol.10 (2), p.313-323 [Periódico revisado por pares]

Oxford: Elsevier Science

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10
1,25-dihydroxyvitamin D as Predictor of Renal Worsening Function in Chronic Kidney Disease. Results From the PASCaL-1,25D Study
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1,25-dihydroxyvitamin D as Predictor of Renal Worsening Function in Chronic Kidney Disease. Results From the PASCaL-1,25D Study

Galassi, Andrea ; Fasulo, Eliana Maria ; Ciceri, Paola ; Casazza, Roberta ; Bonelli, Fabrizio ; Zierold, Claudia ; Calleri, Mariella ; Blocki, Frank A ; Palmieri, Maria Assunta ; Mastronardo, Claudio ; Cozzolino, Mario G

Frontiers in medicine, 2022-03, Vol.9, p.840801-840801 [Periódico revisado por pares]

Switzerland: Frontiers Media S.A

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