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1 |
Material Type: Artigo
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Pyrrole: An emerging scaffold for construction of valuable therapeutic agentsGholap, Somnath S.European journal of medicinal chemistry, 2016-03, Vol.110, p.13-31 [Periódico revisado por pares]France: Elsevier Masson SASTexto completo disponível |
2 |
Material Type: Tese de Doutorado
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Planejamento, síntese e avaliação biológica de derivados pirrólicos com potencial atividade antiinflamatóriaPancote, Camila GarcelBiblioteca Digital de Teses e Dissertações da USP; Universidade de São Paulo; Faculdade de Ciências Farmacêuticas 2009-06-05Acesso online. A biblioteca também possui exemplares impressos. |
3 |
Material Type: Artigo
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Palladium‐Catalyzed Tandem Cyclization of 2‐(2 Ethynylphenyl)acetonitriles and Isocyanides: Access to IndenopyrrolesHui‐Shu Lin ; Yong‐Zhou Pan ; Yu‐Hong Tian ; Ying‐Ming Pan ; Wang, XuAdvanced synthesis & catalysis, 2022-03, Vol.364 (6), p.1117-1121 [Periódico revisado por pares]Heidelberg: Wiley Subscription Services, IncTexto completo disponível |
4 |
Material Type: Artigo
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Futibatinib, an Irreversible FGFR1-4 Inhibitor, in Patients with Advanced Solid Tumors Harboring FGF / FGFR Aberrations: A Phase I Dose-Expansion StudyMeric-Bernstam, Funda ; Bahleda, Rastislav ; Hierro, Cinta ; Sanson, Marc ; Bridgewater, John ; Arkenau, Hendrik-Tobias ; Tran, Ben ; Kelley, Robin Kate ; Park, Joon Oh ; Javle, Milind ; He, Yaohua ; Benhadji, Karim A ; Goyal, LipikaCancer discovery, 2022-02, Vol.12 (2), p.402-415United States: American Association for Cancer ResearchTexto completo disponível |
5 |
Material Type: Artigo
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Safety and efficacy of avapritinib in advanced systemic mastocytosis: the phase 1 EXPLORER trialDeAngelo, Daniel J ; Radia, Deepti H ; George, Tracy I ; Robinson, William A ; Quiery, Albert T ; Drummond, Mark W ; Bose, Prithviraj ; Hexner, Elizabeth O ; Winton, Elliott F ; Horny, Hans-Peter ; Tugnait, Meera ; Schmidt-Kittler, Oleg ; Evans, Erica K ; Lin, Hui-Min ; Mar, Brenton G ; Verstovsek, Srdan ; Deininger, Michael W ; Gotlib, JasonNature medicine, 2021-12, Vol.27 (12), p.2183-2191 [Periódico revisado por pares]United States: Nature Publishing GroupTexto completo disponível |
6 |
Material Type: Artigo
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Silver-Catalyzed Isocyanide-Alkyne Cycloaddition: A General and Practical Method to Oligosubstituted PyrrolesLiu, Jianquan ; Fang, Zhongxue ; Zhang, Qian ; Liu, Qun ; Bi, XiheAngewandte Chemie (International ed.), 2013-07, Vol.52 (27), p.6953-6957 [Periódico revisado por pares]Weinheim: WILEY-VCH VerlagTexto completo disponível |
7 |
Material Type: Artigo
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Discovery of sulfadrug–pyrrole conjugates as carbonic anhydrase and acetylcholinesterase inhibitorsGümüş, Mehmet ; Babacan, Şemsi N. ; Demir, Yeliz ; Sert, Yusuf ; Koca, İrfan ; Gülçin, İlhamiArchiv der Pharmazie (Weinheim), 2022-01, Vol.355 (1), p.e2100242-n/a [Periódico revisado por pares]Germany: Wiley Subscription Services, IncTexto completo disponível |
8 |
Material Type: Artigo
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Identification of N‑{cis-3-[Methyl(7H‑pyrrolo[2,3‑d]pyrimidin-4-yl)amino]cyclobutyl}propane-1-sulfonamide (PF-04965842): A Selective JAK1 Clinical Candidate for the Treatment of Autoimmune DiseasesVazquez, Michael L ; Kaila, Neelu ; Strohbach, Joseph W ; Trzupek, John D ; Brown, Matthew F ; Flanagan, Mark E ; Mitton-Fry, Mark J ; Johnson, Timothy A ; TenBrink, Ruth E ; Arnold, Eric P ; Basak, Arindrajit ; Heasley, Steven E ; Kwon, Soojin ; Langille, Jonathan ; Parikh, Mihir D ; Griffin, Sarah H ; Casavant, Jeffrey M ; Duclos, Brian A ; Fenwick, Ashley E ; Harris, Thomas M ; Han, Seungil ; Caspers, Nicole ; Dowty, Martin E ; Yang, Xin ; Banker, Mary Ellen ; Hegen, Martin ; Symanowicz, Peter T ; Li, Li ; Wang, Lu ; Lin, Tsung H ; Jussif, Jason ; Clark, James D ; Telliez, Jean-Baptiste ; Robinson, Ralph P ; Unwalla, RayJournal of medicinal chemistry, 2018-02, Vol.61 (3), p.1130-1152 [Periódico revisado por pares]United States: American Chemical SocietyTexto completo disponível |
9 |
Material Type: Artigo
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Direct Synthesis of Pyrroles by Dehydrogenative Coupling of β-Aminoalcohols with Secondary Alcohols Catalyzed by Ruthenium Pincer ComplexesSrimani, Dipankar ; Ben-David, Yehoshoa ; Milstein, DavidAngewandte Chemie (International ed.), 2013-04, Vol.52 (14), p.4012-4015 [Periódico revisado por pares]Weinheim: WILEY-VCH VerlagTexto completo disponível |
10 |
Material Type: Artigo
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Discovery of IDO1 inhibitors containing a decahydroquinoline, decahydro-1,6-naphthyridine, or octahydro-1H-pyrrolo[3,2-c]pyridine scaffoldYu, Wensheng ; Deng, Yongqi ; Sloman, David ; Li, Derun ; Liu, Kun ; Fradera, Xavier ; Lesburg, Charles A. ; Martinot, Theo ; Doty, Amy ; Ferguson, Heidi ; Richard Miller, J. ; Knemeyer, Ian ; Otte, Karin ; Vincent, Stella ; Sciammetta, Nunzio ; Jonathan Bennett, David ; Han, YongxinBioorganic & medicinal chemistry letters, 2021-10, Vol.49, p.128314-128314, Article 128314 [Periódico revisado por pares]England: Elsevier LtdTexto completo disponível |