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Preclinical Evaluation of the Effects of Trazpiroben (TAK-906), a Novel, Potent Dopamine D 2 /D 3 Receptor Antagonist for the Management of Gastroparesis
Preclinical Evaluation of the Effects of Trazpiroben (TAK-906), a Novel, Potent Dopamine D 2 /D 3 Receptor Antagonist for the Management of Gastroparesis
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Preclinical Evaluation of the Effects of Trazpiroben (TAK-906), a Novel, Potent Dopamine D 2 /D 3 Receptor Antagonist for the Management of Gastroparesis

Whiting, Roger L ; Choppin, Agnes ; Luehr, Gary ; Jasper, Jeffrey R

The Journal of pharmacology and experimental therapeutics, 2021-10, Vol.379 (1), p.85-95 [Periódico revisado por pares]

United States

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2
Design, Synthesis, and Structure–Activity Relationship Studies of a Series of [4-(4-Carboxamidobutyl)]-1-arylpiperazines: Insights into Structural Features Contributing to Dopamine D3 versus D2 Receptor Subtype Selectivity
Design, Synthesis, and Structure–Activity Relationship Studies of a Series of [4-(4-Carboxamidobutyl)]-1-arylpiperazines: Insights into Structural Features Contributing to Dopamine D3 versus D2 Receptor Subtype Selectivity
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Design, Synthesis, and Structure–Activity Relationship Studies of a Series of [4-(4-Carboxamidobutyl)]-1-arylpiperazines: Insights into Structural Features Contributing to Dopamine D3 versus D2 Receptor Subtype Selectivity

Ananthan, Subramaniam ; Saini, Surendra K ; Zhou, Guangyan ; Hobrath, Judith V ; Padmalayam, Indira ; Zhai, Ling ; Bostwick, J. Robert ; Antonio, Tamara ; Reith, Maarten E. A ; McDowell, Shea ; Cho, Eunie ; McAleer, Leah ; Taylor, Michelle ; Luedtke, Robert R

Journal of medicinal chemistry, 2014-08, Vol.57 (16), p.7042-7060 [Periódico revisado por pares]

United States: American Chemical Society

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3
Structure of the Human Dopamine D3 Receptor in Complex with a D2/D3 Selective Antagonist
Structure of the Human Dopamine D3 Receptor in Complex with a D2/D3 Selective Antagonist
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Structure of the Human Dopamine D3 Receptor in Complex with a D2/D3 Selective Antagonist

Chien, Ellen Y.T ; Liu, Wei ; Zhao, Qiang ; Katritch, Vsevolod ; Won Han, Gye ; Hanson, Michael A ; Shi, Lei ; Newman, Amy Hauck ; Javitch, Jonathan A ; Cherezov, Vadim ; Stevens, Raymond C

Science (American Association for the Advancement of Science), 2010-11, Vol.330 (6007), p.1091-1095 [Periódico revisado por pares]

Washington, DC: American Association for the Advancement of Science

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4
Recent Progress in Development of Dopamine Receptor Subtype-Selective Agents:  Potential Therapeutics for Neurological and Psychiatric Disorders
Recent Progress in Development of Dopamine Receptor Subtype-Selective Agents:  Potential Therapeutics for Neurological and Psychiatric Disorders
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Recent Progress in Development of Dopamine Receptor Subtype-Selective Agents:  Potential Therapeutics for Neurological and Psychiatric Disorders

Zhang, Ao ; Neumeyer, John L. ; Baldessarini, Ross J.

Chemical reviews, 2007-01, Vol.107 (1), p.274-302 [Periódico revisado por pares]

United States: American Chemical Society

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5
Ligand discovery from a dopamine D3 receptor homology model and crystal structure
Ligand discovery from a dopamine D3 receptor homology model and crystal structure
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Ligand discovery from a dopamine D3 receptor homology model and crystal structure

Carlsson, Jens ; Coleman, Ryan G ; Setola, Vincent ; Irwin, John J ; Fan, Hao ; Schlessinger, Avner ; Sali, Andrej ; Roth, Bryan L ; Shoichet, Brian K

Nature chemical biology, 2011-09, Vol.7 (11), p.769-778 [Periódico revisado por pares]

United States: Nature Publishing Group

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6
Highly Selective Dopamine D3 Receptor (D3R) Antagonists and Partial Agonists Based on Eticlopride and the D3R Crystal Structure: New Leads for Opioid Dependence Treatment
Highly Selective Dopamine D3 Receptor (D3R) Antagonists and Partial Agonists Based on Eticlopride and the D3R Crystal Structure: New Leads for Opioid Dependence Treatment
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Highly Selective Dopamine D3 Receptor (D3R) Antagonists and Partial Agonists Based on Eticlopride and the D3R Crystal Structure: New Leads for Opioid Dependence Treatment

Kumar, Vivek ; Bonifazi, Alessandro ; Ellenberger, Michael P ; Keck, Thomas M ; Pommier, Elie ; Rais, Rana ; Slusher, Barbara S ; Gardner, Eliot ; You, Zhi-Bing ; Xi, Zheng-Xiong ; Newman, Amy Hauck

Journal of medicinal chemistry, 2016-08, Vol.59 (16), p.7634-7650 [Periódico revisado por pares]

United States: American Chemical Society

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7
Design and Mechanism of (S)‑3-Amino-4-(difluoromethylenyl)cyclopent-1-ene-1-carboxylic Acid, a Highly Potent γ‑Aminobutyric Acid Aminotransferase Inactivator for the Treatment of Addiction
Design and Mechanism of (S)‑3-Amino-4-(difluoromethylenyl)cyclopent-1-ene-1-carboxylic Acid, a Highly Potent γ‑Aminobutyric Acid Aminotransferase Inactivator for the Treatment of Addiction
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Design and Mechanism of (S)‑3-Amino-4-(difluoromethylenyl)cyclopent-1-ene-1-carboxylic Acid, a Highly Potent γ‑Aminobutyric Acid Aminotransferase Inactivator for the Treatment of Addiction

Juncosa, Jose I ; Takaya, Kenji ; Le, Hoang V ; Moschitto, Matthew J ; Weerawarna, Pathum M ; Mascarenhas, Romila ; Liu, Dali ; Dewey, Stephen L ; Silverman, Richard B

Journal of the American Chemical Society, 2018-02, Vol.140 (6), p.2151-2164 [Periódico revisado por pares]

United States: American Chemical Society

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8
Medication discovery for addiction: Translating the dopamine D3 receptor hypothesis
Medication discovery for addiction: Translating the dopamine D3 receptor hypothesis
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Medication discovery for addiction: Translating the dopamine D3 receptor hypothesis

Newman, Amy Hauck ; Blaylock, Brandi L. ; Nader, Michael A. ; Bergman, Jack ; Sibley, David R. ; Skolnick, Phil

Biochemical pharmacology, 2012-10, Vol.84 (7), p.882-890 [Periódico revisado por pares]

England: Elsevier Inc

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9
Discovery and characterization of benzyloxy piperidine based dopamine 4 receptor antagonists
Discovery and characterization of benzyloxy piperidine based dopamine 4 receptor antagonists
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Discovery and characterization of benzyloxy piperidine based dopamine 4 receptor antagonists

Tolentino, Kirsten T. ; Mashinson, Viktoriya ; Vadukoot, Anish K. ; Hopkins, Corey R.

Bioorganic & medicinal chemistry letters, 2022-04, Vol.61, p.128615-128615, Article 128615 [Periódico revisado por pares]

England: Elsevier Ltd

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10
Distinct inactive conformations of the dopamine D2 and D3 receptors correspond to different extents of inverse agonism
Distinct inactive conformations of the dopamine D2 and D3 receptors correspond to different extents of inverse agonism
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Distinct inactive conformations of the dopamine D2 and D3 receptors correspond to different extents of inverse agonism

Lane, J Robert ; Abramyan, Ara M ; Adhikari, Pramisha ; Keen, Alastair C ; Lee, Kuo-Hao ; Sanchez, Julie ; Verma, Ravi Kumar ; Lim, Herman D ; Yano, Hideaki ; Javitch, Jonathan A ; Shi, Lei

eLife, 2020-01, Vol.9 [Periódico revisado por pares]

England: eLife Science Publications, Ltd

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