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1 |
Material Type: Artigo
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Functional Pyrazolo[1,5- a ]pyrimidines: Current Approaches in Synthetic Transformations and Uses As an Antitumor ScaffoldArias-Gómez, Andres ; Godoy, Andrés ; Portilla, JaimeMolecules (Basel, Switzerland), 2021-05, Vol.26 (9), p.2708 [Periódico revisado por pares]Switzerland: MDPI AGTexto completo disponível |
2 |
Material Type: Artigo
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Thieno[2,3-d]pyrimidine as a promising scaffold in medicinal chemistry: Recent advancesAli, Eslam M.H. ; Abdel-Maksoud, Mohammed S. ; Oh, Chang-HyunBioorganic & medicinal chemistry, 2019-04, Vol.27 (7), p.1159-1194 [Periódico revisado por pares]England: Elsevier LtdTexto completo disponível |
3 |
Material Type: Artigo
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Design and Synthesis of New Thiophene/Thieno[2,3- d ]pyrimidines along with Their Cytotoxic Biological Evaluation as Tyrosine Kinase Inhibitors in Addition to Their Apoptotic and Autophagic InductionElmongy, Elshaymaa I ; Attallah, Nashwah G M ; Altwaijry, Najla ; AlKahtani, Manal Mubarak ; Henidi, Hanan AliMolecules (Basel, Switzerland), 2021-12, Vol.27 (1), p.123 [Periódico revisado por pares]Switzerland: MDPI AGTexto completo disponível |
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Material Type: Artigo
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Heterocyclic steroids: Efficient routes for annulation of pentacyclic steroidal pyrimidinesMonier, M. ; El-Mekabaty, Ahmed ; Abdel-Latif, Doaa ; Doğru Mert, Başak ; Elattar, Khaled M.Steroids, 2020-02, Vol.154, p.108548-108548, Article 108548 [Periódico revisado por pares]United States: Elsevier IncTexto completo disponível |
5 |
Material Type: Artigo
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Synthesis of a new series of pyrazolo[1,5-a]pyrimidines as CDK2 inhibitors and anti-leukemiaAlmehmadi, Samar J. ; Alsaedi, Amani M.R. ; Harras, Marwa F. ; Farghaly, Thoraya A.Bioorganic chemistry, 2021-12, Vol.117, p.105431-105431, Article 105431 [Periódico revisado por pares]United States: Elsevier IncTexto completo disponível |
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Material Type: Artigo
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Novel pyrazolo[3,4-d]pyrimidines: design, synthesis, anticancer activity, dual EGFR/ErbB2 receptor tyrosine kinases inhibitory activity, effects on cell cycle profile and caspase-3-mediated apoptosisMaher, Mai ; Kassab, Asmaa E. ; Zaher, Ashraf F. ; Mahmoud, ZeinabJournal of enzyme inhibition and medicinal chemistry, 2019-01, Vol.34 (1), p.532-546 [Periódico revisado por pares]England: Taylor & FrancisTexto completo disponível |
7 |
Material Type: Artigo
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New pyrimidine and pyrazole-based compounds as potential EGFR inhibitors: Synthesis, anticancer, antimicrobial evaluation and computational studiesOthman, Ismail M.M. ; Alamshany, Zahra M. ; Tashkandi, Nada Y. ; Gad-Elkareem, Mohamed A.M. ; Anwar, Manal M. ; Nossier, Eman S.Bioorganic chemistry, 2021-09, Vol.114, p.105078, Article 105078 [Periódico revisado por pares]United States: Elsevier IncTexto completo disponível |
8 |
Material Type: Artigo
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Design, synthesis, molecular docking and in silico ADMET profile of pyrano[2,3-d]pyrimidine derivatives as antimicrobial and anticancer agentsAbd El-Sattar, Nour E.A. ; El‐Adl, Khaled ; El-Hashash, Maher A. ; Salama, Samir A. ; Elhady, Mostafa M.Bioorganic chemistry, 2021-10, Vol.115, p.105186-105186, Article 105186 [Periódico revisado por pares]United States: Elsevier IncTexto completo disponível |
9 |
Material Type: Artigo
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Synthesis and in vitro antitumor evaluation of some new thiophenes and thieno[2,3-d]pyrimidine derivativesFouad, Mahasen M. ; El-Bendary, Eman R. ; suddek, Ghada M. ; Shehata, Ihsan A. ; El-Kerdawy, Mohamed M.Bioorganic chemistry, 2018-12, Vol.81, p.587-598 [Periódico revisado por pares]United States: Elsevier IncTexto completo disponível |
10 |
Material Type: Artigo
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Design and synthesis of pyrazolo[3,4-d]pyrimidines: Nitric oxide releasing compounds targeting hepatocellular carcinomaElshaier, Yaseen A.M.M. ; Shaaban, Mohamed A. ; Abd El Hamid, Mohammed K. ; Abdelrahman, Mostafa H. ; Abou-Salim, Mahrous A. ; Elgazwi, Sara M. ; Halaweish, FathiBioorganic & medicinal chemistry, 2017-06, Vol.25 (12), p.2956-2970 [Periódico revisado por pares]England: Elsevier LtdTexto completo disponível |