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1 |
Material Type: Article
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Chemoproteomic Profiling of Itaconation by Bioorthogonal Probes in Inflammatory MacrophagesQin, Wei ; Zhang, Yanling ; Tang, Huan ; Liu, Dongyang ; Chen, Ying ; Liu, Yuan ; Wang, ChuJournal of the American Chemical Society, 2020-06, Vol.142 (25), p.10894-10898 [Peer Reviewed Journal]United States: American Chemical SocietyFull text available |
2 |
Material Type: Article
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Dipropargyl substituted diphenylpyrimidines as dual inhibitors of monoamine oxidase and acetylcholinesteraseKumar, Bhupinder ; Kumar, Vijay ; Prashar, Vikash ; Saini, Suresh ; Dwivedi, Ashish Ranjan ; Bajaj, Beenu ; Mehta, Devashish ; Parkash, Jyoti ; Kumar, VinodEuropean journal of medicinal chemistry, 2019-09, Vol.177, p.221-234 [Peer Reviewed Journal]France: Elsevier Masson SASFull text available |
3 |
Material Type: Article
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High-Affinity Alkynyl Bisubstrate Inhibitors of Nicotinamide N‑Methyltransferase (NNMT)Policarpo, Rocco L ; Decultot, Ludovic ; May, Elizabeth ; Kuzmič, Petr ; Carlson, Samuel ; Huang, Danny ; Chu, Vincent ; Wright, Brandon A ; Dhakshinamoorthy, Saravanakumar ; Kannt, Aimo ; Rani, Shilpa ; Dittakavi, Sreekanth ; Panarese, Joseph D ; Gaudet, Rachelle ; Shair, Matthew DJournal of medicinal chemistry, 2019-11, Vol.62 (21), p.9837-9873 [Peer Reviewed Journal]United States: American Chemical SocietyFull text available |
4 |
Material Type: Article
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Azide-alkyne cycloaddition towards 1H-1,2,3-triazole-tethered gatifloxacin and isatin conjugates: Design, synthesis and in vitro anti-mycobacterial evaluationXu, Zhi ; Song, Xu-Feng ; Hu, Yuan-Qiang ; Qiang, Min ; Lv, Zao-ShengEuropean journal of medicinal chemistry, 2017-09, Vol.138, p.66-71 [Peer Reviewed Journal]France: Elsevier Masson SASFull text available |
5 |
Material Type: Article
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Systemic HIV and SIV latency reversal via non-canonical NF-κB signalling in vivoNixon, Christopher C ; Mavigner, Maud ; Sampey, Gavin C ; Brooks, Alyssa D ; Spagnuolo, Rae Ann ; Irlbeck, David M ; Mattingly, Cameron ; Ho, Phong T ; Schoof, Nils ; Cammon, Corinne G ; Tharp, Greg K ; Kanke, Matthew ; Wang, Zhang ; Cleary, Rachel A ; Upadhyay, Amit A ; De, Chandrav ; Wills, Saintedym R ; Falcinelli, Shane D ; Galardi, Cristin ; Walum, Hasse ; Schramm, Nathaniel J ; Deutsch, Jennifer ; Lifson, Jeffrey D ; Fennessey, Christine M ; Keele, Brandon F ; Jean, Sherrie ; Maguire, Sean ; Liao, Baolin ; Browne, Edward P ; Ferris, Robert G ; Brehm, Jessica H ; Favre, David ; Vanderford, Thomas H ; Bosinger, Steven E ; Jones, Corbin D ; Routy, Jean-Pierre ; Archin, Nancie M ; Margolis, David M ; Wahl, Angela ; Dunham, Richard M ; Silvestri, Guido ; Chahroudi, Ann ; Garcia, J VictorNature (London), 2020-02, Vol.578 (7793), p.160-165 [Peer Reviewed Journal]England: Nature Publishing GroupFull text available |
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Material Type: Article
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Alkyne as a Latent Warhead to Covalently Target SARS-CoV‑2 Main ProteaseNgo, Chau ; Fried, William ; Aliyari, Saba ; Feng, Joshua ; Qin, Chao ; Zhang, Shilei ; Yang, Hanjing ; Shanaa, Jean ; Feng, Pinghui ; Cheng, Genhong ; Chen, Xiaojiang S. ; Zhang, ChaoJournal of medicinal chemistry, 2023-09, Vol.66 (17), p.12237-12248 [Peer Reviewed Journal]United States: American Chemical SocietyFull text available |
7 |
Material Type: Article
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Phthalocyanine–Peptide Conjugates: Receptor-Targeting Bifunctional Agents for Imaging and Photodynamic TherapyRanyuk, Elena ; Cauchon, Nicole ; Klarskov, Klaus ; Guérin, Brigitte ; van Lier, Johan EJournal of medicinal chemistry, 2013-02, Vol.56 (4), p.1520-1534 [Peer Reviewed Journal]United States: American Chemical SocietyFull text available |
8 |
Material Type: Article
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CARD8 is an inflammasome sensor for HIV-1 protease activityWang, Qiankun ; Gao, Hongbo ; Clark, Kolin M ; Mugisha, Christian Shema ; Davis, Keanu ; Tang, Jack P ; Harlan, Gray H ; DeSelm, Carl J ; Presti, Rachel M ; Kutluay, Sebla B ; Shan, LiangScience (American Association for the Advancement of Science), 2021-03, Vol.371 (6535), p.1224 [Peer Reviewed Journal]United States: American Association for the Advancement of ScienceFull text available |
9 |
Material Type: Article
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Efficacy and effect on lipid profiles of switching to ainuovirine-based regimen versus continuing efavirenz-based regimen in people with HIV-1: 24-week results from a real-world, retrospective, multi-center cohort studyWang, Chunmei ; Yu, Xiaoli ; Ke, Yingchun ; Fu, Yanhua ; Luo, Yanhe ; Li, Ying ; Bi, Yanmei ; Chen, Xingqiong ; Li, Linghua ; Zhao, Xiuhong ; Chen, Zhong Martinez, Miguel AngelAntimicrobial agents and chemotherapy, 2024-04, Vol.68 (4), p.e0166823-e0166823 [Peer Reviewed Journal]United States: American Society for MicrobiologyFull text available |
10 |
Material Type: Article
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An Alkynylpyrimidine-Based Covalent Inhibitor That Targets a Unique Cysteine in NF-κB-Inducing KinaseAl-Khawaldeh, Islam ; Al Yasiri, Mohammed J ; Aldred, Gregory G ; Basmadjian, Christine ; Bordoni, Cinzia ; Harnor, Suzannah J ; Heptinstall, Amy B ; Hobson, Stephen J ; Jennings, Claire E ; Khalifa, Shaimaa ; Lebraud, Honorine ; Martin, Mathew P ; Miller, Duncan C ; Shrives, Harry J ; de Souza, João V ; Stewart, Hannah L ; Temple, Max ; Thomas, Huw D ; Totobenazara, Jane ; Tucker, Julie A ; Tudhope, Susan J ; Wang, Lan Z ; Bronowska, Agnieszka K ; Cano, Céline ; Endicott, Jane A ; Golding, Bernard T ; Hardcastle, Ian R ; Hickson, Ian ; Wedge, Stephen R ; Willmore, Elaine ; Noble, Martin E. M ; Waring, Michael JJournal of medicinal chemistry, 2021-07, Vol.64 (14), p.10001-10018 [Peer Reviewed Journal]United States: American Chemical SocietyFull text available |