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Refinado por: Nome da Publicação: Bioorganic & Medicinal Chemistry Letters remover
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1
Stereochemical properties of quazepam and its affinity for the GABAA receptor
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Stereochemical properties of quazepam and its affinity for the GABAA receptor

Takano, Ryota ; Tanaka, Ryoko ; Nakamura, Kayo ; Tabata, Hidetsugu ; Oshitari, Tetsuta ; Natsugari, Hideaki ; Takahashi, Hideyo

Bioorganic & medicinal chemistry letters, 2024-09, Vol.110, p.129854, Article 129854 [Periódico revisado por pares]

Elsevier Ltd

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2
Ophiobolin A derivatives with enhanced activities under tumor-relevant acidic conditions
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Artigo
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Ophiobolin A derivatives with enhanced activities under tumor-relevant acidic conditions

Maslivetc, Vladimir A. ; Nabiul Hasan, Md ; Boari, Angela ; Zejnelovski, Arben ; Evidente, Antonio ; Sun, Dandan ; Kornienko, Alexander

Bioorganic & medicinal chemistry letters, 2024-09, Vol.110, p.129863, Article 129863 [Periódico revisado por pares]

Elsevier Ltd

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3
[1,2,4]Triazolo[1,5-a]pyrimidine derivatives: Structure-activity relationship study leading to highly selective ENPP1 inhibitors
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[1,2,4]Triazolo[1,5-a]pyrimidine derivatives: Structure-activity relationship study leading to highly selective ENPP1 inhibitors

Kawaguchi, Mitsuyasu ; Minami, Shohei ; Ieda, Naoya ; Nakagawa, Hidehiko

Bioorganic & medicinal chemistry letters, 2024-09, Vol.110, p.129820, Article 129820 [Periódico revisado por pares]

Elsevier Ltd

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4
Extended voltage imaging in cardiomyocytes with a triplet state quencher-stabilized silicon rhodamine
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Extended voltage imaging in cardiomyocytes with a triplet state quencher-stabilized silicon rhodamine

Martinez, Kayli N. ; Gerstner, Nels C. ; Yang, Samantha J. ; Miller, Evan W.

Bioorganic & medicinal chemistry letters, 2024-09, Vol.109 (C), p.129842, Article 129842 [Periódico revisado por pares]

United Kingdom: Elsevier Ltd

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5
PEG-lipid-modified agonistic antibody against tumor necrosis factor receptor family elicits superior apoptosis-inducing activity against human carcinoma
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PEG-lipid-modified agonistic antibody against tumor necrosis factor receptor family elicits superior apoptosis-inducing activity against human carcinoma

Niwa, Takako ; Kasuya, Yuji ; Ichikawa, Kimihisa ; Yoshida, Hiroko ; Kurimoto, Akiko ; Tanaka, Kento ; Morita, Koji

Bioorganic & medicinal chemistry letters, 2024-09, Vol.109, p.129840, Article 129840 [Periódico revisado por pares]

Elsevier Ltd

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6
Michael addition-activated alkylation of G-quadruplex DNA with methylamine-protected vinyl-quinazolinone derivatives
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Michael addition-activated alkylation of G-quadruplex DNA with methylamine-protected vinyl-quinazolinone derivatives

Chen, Yutong ; Onizuka, Kazumitsu ; Nagatsugi, Fumi

Bioorganic & medicinal chemistry letters, 2024-09, Vol.109, p.129855, Article 129855 [Periódico revisado por pares]

Elsevier Ltd

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7
Key challenges in TB drug discovery: A perspective
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Key challenges in TB drug discovery: A perspective

Shaik, Baji Baba ; Karpoormath, Rajshekhar

Bioorganic & medicinal chemistry letters, 2024-09, Vol.109, p.129846, Article 129846 [Periódico revisado por pares]

Elsevier Ltd

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8
Detecting 2′-5′-adenosine linked nucleic acids via acylation of secondary hydroxy functionality
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Detecting 2′-5′-adenosine linked nucleic acids via acylation of secondary hydroxy functionality

Chen, Xiaoqian ; Guo, Yuyang ; Wang, Rui

Bioorganic & medicinal chemistry letters, 2024-09, Vol.109, p.129847, Article 129847 [Periódico revisado por pares]

Elsevier Ltd

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9
Novel 4-[4-(4-methylpiperazin-1-yl)phenyl]-6-arylpyrimidine derivatives and their antitrypanosomal activities against T.brucei
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Novel 4-[4-(4-methylpiperazin-1-yl)phenyl]-6-arylpyrimidine derivatives and their antitrypanosomal activities against T.brucei

Taylor, Annie E. ; Hering, Moritz ; Elsegood, Mark R.J. ; Teat, Simon J. ; Weaver, George W. ; Arroo, Randolph R.J. ; Kaiser, Marcel ; Maeser, Pascal ; Bhambra, Avninder S.

Bioorganic & medicinal chemistry letters, 2024-09, Vol.109 (C), p.129825, Article 129825 [Periódico revisado por pares]

England: Elsevier Ltd

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10
Design and synthesis of novel fluorene derivatives as inhibitors of pyruvate dehydrogenase kinase
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Design and synthesis of novel fluorene derivatives as inhibitors of pyruvate dehydrogenase kinase

Inoue, Masafumi ; Nagamori, Hironobu ; Morita, Toru ; Kobayashi, Satoru ; Suzawa, Koichi ; Kitao, Yuki ; Saito, Tomoyuki ; Kawahara, Iichiro ; Orita, Takuya ; Akai, Shota ; Adachi, Tsuyoshi ; Motomura, Takahisa

Bioorganic & medicinal chemistry letters, 2024-09, Vol.109, p.129839, Article 129839 [Periódico revisado por pares]

Elsevier Ltd

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