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Material Type: Artículo
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1-[1-(2-Benzo[b]thiopheneyl)cyclohexyl]piperidine Hydrochloride (BTCP) Yields Two Active Primary Metabolites in Vitro: Synthesis, Identification from Rat Liver Microsome Extracts, and Affinity for the Neuronal Dopamine TransporterDeleuze-Masquefa, Carine ; Michaud, Martine ; Vignon, Jacques ; Kamenka, Jean-MarcJournal of medicinal chemistry, 1997-12, Vol.40 (25), p.4019-4025 [Revista revisada por pares]Washington, DC: American Chemical SocietyTexto completo disponible |
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Material Type: Artículo
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1-(1-Naphthyl)piperazine as a novel template for 5-HT6 serotonin receptor ligandsLEE, Mase ; RANGISETTY, Jagadeesh B ; PULLAGURLA, Manik R ; DUKAT, Małgorzata ; SETOLA, Vince ; ROTH, Bryan L ; GLENNON, Richard ABioorganic & medicinal chemistry letters, 2005-03, Vol.15 (6), p.1707-1711 [Revista revisada por pares]Oxford: ElsevierTexto completo disponible |
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Material Type: Artículo
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1-(1,2,5-Thiadiazol-4-yl)-4-azatricyclo[2.2.1.02,6]heptanes as New Potent Muscarinic M1 Agonists: Structure−Activity Relationship for 3-Aryl-2-propyn-1-yloxy and 3-Aryl-2-propyn-1-ylthio DerivativesJeppesen, Lone ; Olesen, Preben H ; Hansen, Lena ; Sheardown, Malcolm J ; Thomsen, Christian ; Rasmussen, Thøger ; Jensen, Anders Fink ; Christensen, Michael S ; Rimvall, Karin ; Ward, John S ; Whitesitt, Celia ; Calligaro, David O ; Bymaster, Frank P ; Delapp, Neil W ; Felder, Christian C ; Shannon, Harlan E ; Sauerberg, PerJournal of medicinal chemistry, 1999-06, Vol.42 (11), p.1999-2006 [Revista revisada por pares]Washington, DC: American Chemical SocietyTexto completo disponible |
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Material Type: Artículo
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1, 2, 4-Triazine N-oxide Derivatives: Studies as Potential Hypoxic Cytotoxins. Part IICerecetto, Hugo ; González, Mercedes ; Onetto, Silvia ; Saenz, Patricia ; Ezpeleta, Olga ; de Ceráin, Adela López ; Monge, AntonioArchiv der Pharmazie (Weinheim), 2004-05, Vol.337 (5), p.247-258 [Revista revisada por pares]Weinheim: WILEY-VCH VerlagTexto completo disponible |
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Material Type: Artículo
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1, 2, 4-Triazine N-oxide Derivatives: Studies as Potential Hypoxic Cytotoxins. Part IIICerecetto, Hugo ; González, Mercedes ; Risso, Mariela ; Saenz, Patricia ; Olea-Azar, Claudio ; Bruno, Ana M. ; Azqueta, Amaia ; de Ceráin, Adela López ; Monge, AntonioArchiv der Pharmazie (Weinheim), 2004-05, Vol.337 (5), p.271-280 [Revista revisada por pares]Weinheim: WILEY-VCH VerlagTexto completo disponible |
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Material Type: Artículo
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1,1-Bis(3′-indolyl)-1-(p-substituted phenyl)methanes inhibit colon cancer cell and tumor growth through activation of c-jun N-terminal kinaseLei, Ping ; Abdelrahim, Maen ; Cho, Sung Dae ; Liu, Shengxi ; Chintharlapalli, Sudhakar ; Safe, StephenCarcinogenesis (New York), 2008-06, Vol.29 (6), p.1139-1147 [Revista revisada por pares]Oxford: Oxford University PressTexto completo disponible |
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Material Type: Artículo
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1,1-Diarylalkenes as anticancer agents: Dual inhibitors of tubulin polymerization and phosphodiesterase 4Ruchelman, Alexander L. ; Man, Hon-Wah ; Chen, Roger ; Liu, Wei ; Lu, Ling ; Cedzik, Dorota ; Zhang, Ling ; Leisten, Jim ; Collette, Alice ; Narla, Rama Krishna ; Raymon, Heather K. ; Muller, George W.Bioorganic & medicinal chemistry, 2011-11, Vol.19 (21), p.6356-6374 [Revista revisada por pares]Amsterdam: Elsevier LtdTexto completo disponible |
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Material Type: Artículo
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1,1-Diphenyl-2-picrylhydrazyl radical-scavenging compounds from soybean miso and antiproliferative activity of isoflavones from soybean miso toward the cancer cell linesHirota, A. (Shizuoka Univ. (Japan)) ; Taki, S ; Kawaii, S ; Yano, M ; Abe, NBioscience, biotechnology, and biochemistry, 2000-05, Vol.64 (5), p.1038-1040 [Revista revisada por pares]Tokyo: Japan Society for Bioscience, Biotechnology, and AgrochemistryTexto completo disponible |
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Material Type: Artículo
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1,12-Substituted tetracyclines as antioxidant agentsLertvorachon, Jittiwud ; Kim, Jong-Pyung ; Soldatov, Dmitriy V. ; Boyd, Jason ; Roman, Gheorghe ; Cho, Sung Ju ; Popek, Tomasz ; Jung, Young-Sik ; Lau, Peter C.K. ; Konishi, YasuoBioorganic & medicinal chemistry, 2005-08, Vol.13 (15), p.4627-4637 [Revista revisada por pares]Oxford: Elsevier LtdTexto completo disponible |
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Material Type: Artículo
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1,1,3-Trioxo-2H,4H-Thieno[3,4-e][1,2,4]Thiadiazine (TTD) Derivatives: a New Class of Nonnucleoside Human Immunodeficiency Virus Type 1 (HIV-1) Reverse Transcriptase Inhibitors with Anti-HIV-1 ActivityWITVROUW, M ; ARRANZ, M. E ; ESNOUF, R ; VAN MEERVELT, L ; VEGA, S ; BALZARINI, J ; DE CLERCQ, E ; PANNECOUQUE, C ; DECLERCQ, R ; JONCKHEERE, H ; SCHMIT, J.-C ; VANDAMME, A.-M ; DIAZ, J. A ; INGATE, S. T ; DESMYTER, JAntimicrobial Agents and Chemotherapy, 1998-03, Vol.42 (3), p.618-623 [Revista revisada por pares]Washington, DC: American Society for MicrobiologyTexto completo disponible |