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Material Type: Artigo
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1-(1H-Indol-3-yl)ethanamine Derivatives as Potent Staphylococcus aureus NorA Efflux Pump InhibitorsHequet, Arnaud ; Burchak, Olga N. ; Jeanty, Matthieu ; Guinchard, Xavier ; Le Pihive, Emmanuelle ; Maigre, Laure ; Bouhours, Pascale ; Schneider, Dominique ; Maurin, Max ; Paris, Jean-Marc ; Denis, Jean-Noël ; Jolivalt, ClaudeChemMedChem, 2014-07, Vol.9 (7), p.1534-1545 [Periódico revisado por pares]Weinheim: WILEY-VCH VerlagTexto completo disponível |
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Material Type: Artigo
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1-[2-(1-Cyclobutylpiperidin-4-yloxy)-6,7-dihydro-4H-thiazolo[5,4-c]pyridin-5-yl]propan-1-one: a Histamine H 3 Receptor Inverse Agonist with Efficacy in Animal Models of CognitionShinde, Anil Karbhari ; Badange, Rajesh Kumar ; Reballi, Veena ; Achanta, Pramod Kumar ; Bojja, Kumar ; Manchineella, Sravanthi ; Rao Muddana, Nageswara ; Subramanian, Ramkumar ; Choudary Palacharla, Raghava ; Benade, Vijay ; Jayarajan, Pradeep ; Thentu, Jagadeesh Babu ; Lingavarapu, Bujji Babu ; Yarra, Sivasekhar ; Kagita, Narendra ; Rao Doguparthi, Mallikarjuna ; Mohammed, Abdul Rasheed ; Nirogi, RamakrishnaChemMedChem, 2022-02, Vol.17 (3), p.e202100583 [Periódico revisado por pares]GermanyTexto completo disponível |
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Material Type: Artigo
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1, 2, 4-Triazine N-oxide Derivatives: Studies as Potential Hypoxic Cytotoxins. Part IICerecetto, Hugo ; González, Mercedes ; Onetto, Silvia ; Saenz, Patricia ; Ezpeleta, Olga ; de Ceráin, Adela López ; Monge, AntonioArchiv der Pharmazie (Weinheim), 2004-05, Vol.337 (5), p.247-258 [Periódico revisado por pares]Weinheim: WILEY-VCH VerlagTexto completo disponível |
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Material Type: Artigo
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1, 2, 4-Triazine N-oxide Derivatives: Studies as Potential Hypoxic Cytotoxins. Part IIICerecetto, Hugo ; González, Mercedes ; Risso, Mariela ; Saenz, Patricia ; Olea-Azar, Claudio ; Bruno, Ana M. ; Azqueta, Amaia ; de Ceráin, Adela López ; Monge, AntonioArchiv der Pharmazie (Weinheim), 2004-05, Vol.337 (5), p.271-280 [Periódico revisado por pares]Weinheim: WILEY-VCH VerlagTexto completo disponível |
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Material Type: Artigo
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1‐[(2,3‐Dihydro‐1‐benzofuran‐2‐yl) methyl]piperazines as novel anti‐inflammatory compounds: Synthesis and evaluation on H3R/H4RCorrêa, Michelle Fidelis ; Varela, Marina Themoteo ; Balbino, Aleksandro Martins ; Torrecilhas, Ana Claudia ; Landgraf, Richardt Gama ; Troncone, Lanfranco Ranieri Paolo ; Fernandes, João Paulo dos SantosChemical biology & drug design, 2017-08, Vol.90 (2), p.317-322 [Periódico revisado por pares]Texto completo disponível |
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Material Type: Artigo
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1,2,3-Triazole as a Peptide Surrogate in the Rapid Synthesis of HIV-1 Protease InhibitorsBrik, Ashraf ; Alexandratos, Jerry ; Lin, Ying-Chuan ; Elder, John H ; Olson, Arthur J ; Wlodawer, Alexander ; Goodsell, David S ; Wong, Chi-HueyChembiochem : a European journal of chemical biology, 2005-07, Vol.6 (7), p.1167-1169 [Periódico revisado por pares]Weinheim: Wiley-VCH VerlagTexto completo disponível |
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Material Type: Artigo
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1,2,3‐Triazole‐based esters and carboxylic acids as nonclassical carbonic anhydrase inhibitors capable of cathepsin B inhibitionSiwach, Kiran ; Rani, Manishita ; Vats, Lalit ; Giovannuzzi, Simone ; Paul, Avijit Kumar ; Brahma, Mettle ; Kumari, Neetu ; Maruthi, Mulaka ; Raghav, Neera ; Supuran, Claudiu T. ; Sharma, Pawan K.Archiv der Pharmazie (Weinheim), 2024-03, Vol.357 (3), p.e2300372-n/a [Periódico revisado por pares]Germany: Wiley Subscription Services, IncTexto completo disponível |
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Material Type: Artigo
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1,2,3‐Triazole hybrids as anticancer agents: A reviewAlam, Mohammad MahboobArchiv der Pharmazie (Weinheim), 2022-01, Vol.355 (1), p.e2100158-n/a [Periódico revisado por pares]Germany: Wiley Subscription Services, IncTexto completo disponível |
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Material Type: Artigo
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1,2,3‐Triazole hybrids with anti‐HIV‐1 activityFeng, Lian‐Shun ; Zheng, Man‐Jie ; Zhao, Feng ; Liu, DuanArchiv der Pharmazie (Weinheim), 2021-01, Vol.354 (1), p.e2000163-n/a [Periódico revisado por pares]Germany: Wiley Subscription Services, IncTexto completo disponível |
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Material Type: Artigo
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1,2,3‐Triazole‐linked 5‐benzylidene (thio)barbiturates as novel tyrosinase inhibitors and free‐radical scavengersRanjbar, Sara ; Shahvaran, Parisa‐sadat ; Edraki, Najmeh ; Khoshneviszadeh, Mahsima ; Darroudi, Mahdieh ; Sarrafi, Yaghoub ; Hamzehloueian, Mahshid ; Khoshneviszadeh, MehdiArchiv der Pharmazie (Weinheim), 2020-10, Vol.353 (10), p.e2000058-n/a [Periódico revisado por pares]Frankfurt: Wiley Subscription Services, IncTexto completo disponível |