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1 |
Material Type: Artigo
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1-(2-(2,2,2-trifluoroethoxy)ethyl-1H-pyrazolo[4,3-d]pyrimidines as potent phosphodiesterase 5 (PDE5) inhibitorsTollefson, Michael B ; Acker, Brad A ; Jacobsen, E J ; Hughes, Robert O ; Walker, John K ; Fox, David N A ; Palmer, Michael J ; Freeman, Sandra K ; Yu, Ying ; Bond, Brian RBioorganic & medicinal chemistry letters, 2010-05, Vol.20 (10), p.3125-3128 [Periódico revisado por pares]EnglandTexto completo disponível |
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Material Type: Artigo
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1-(2-Ethoxyethyl)-1H-pyrazolo[4,3-d]pyrimidines as potent phosphodiesterase 5 (PDE5) inhibitorsTOLLEFSON, Michael B ; ACKER, Brad A ; JACOBSEN, E. J ; HUGHES, Robert O ; WALKER, John K ; FOX, David N. A ; PALMER, Michael J ; FREEMAN, Sandra K ; YING YU ; BOND, Brian RBioorganic & medicinal chemistry letters, 2010-05, Vol.20 (10), p.3120-3124 [Periódico revisado por pares]Amsterdam: ElsevierTexto completo disponível |
3 |
Material Type: Artigo
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1-Benzyl derivatives of 5-(arylamino)uracils as anti-HIV-1 and anti-EBV agentsNovikov, Mikhail S. ; Buckheit, Robert W. ; Temburnikar, Kartik ; Khandazhinskaya, Anastasia L. ; Ivanov, Alexander V. ; Seley-Radtke, Katherine L.Bioorganic & medicinal chemistry, 2010-12, Vol.18 (23), p.8310-8314 [Periódico revisado por pares]England: Elsevier LtdTexto completo disponível |
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Material Type: Artigo
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1,1'-(3-methyl-4-phenylthieno[2,3-b]thiophene-2,5-diyl)diethanone as a building block in heterocyclic synthesis. Novel synthesis of some pyrazole and pyrimidine derivativesMabkhot, Yahia Nasser ; Al-Majid, Abdullah Mohammed ; Barakat, Assem ; Alshahrani, Saeed ; Siddiqui, YaminMolecules (Basel, Switzerland), 2011-08, Vol.16 (8), p.6502-6511 [Periódico revisado por pares]Switzerland: MDPI AGTexto completo disponível |
5 |
Material Type: Artigo
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1,2,3,4-Tetrahydro-2-thioxopyrimidine analogs of combretastatin-A4Lee, Lauren ; Davis, Ryan ; Vanderham, Jenna ; Hills, Patrice ; Mackay, Hilary ; Brown, Toni ; Mooberry, Susan L. ; Lee, MosesEuropean journal of medicinal chemistry, 2008-09, Vol.43 (9), p.2011-2015 [Periódico revisado por pares]Oxford: Elsevier Masson SASTexto completo disponível |
6 |
Material Type: Artigo
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18F-labeled pyrazolo[1,5-a]pyrimidine derivatives: synthesis from 2,4-dinitrobenzamide and tosylate precursors and comparative biological evaluation for tumor imaging with positron emission tomographyXu, Jingli ; Liu, Hang ; Li, Guixia ; He, Yong ; Ding, Rui ; Wang, Xiao ; Feng, Man ; Zhang, Shuting ; Chen, Yurong ; Li, Shilei ; Zhao, Mingxia ; Li, Yingruo ; Qi, Chuanmin ; Dang, YonghongMolecules (Basel, Switzerland), 2012-03, Vol.17 (4), p.3774-3793 [Periódico revisado por pares]Switzerland: MDPI AGTexto completo disponível |
7 |
Material Type: Artigo
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(1)H,(13)C and (19)F NMR data of N-substituted 6-(4-methoxyphenyl)-7H-pyrrolo[2,3-d]pyrimidin-4-amines in DMSO-d(6)Sørum, Christopher ; Simić, Nebojsa ; Sundby, Eirik ; Hoff, Bård HelgeMagnetic resonance in chemistry, 2010-03, Vol.48 (3), p.244-248 [Periódico revisado por pares]EnglandTexto completo disponível |
8 |
Material Type: Artigo
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[2 + 2] Photocycloaddition Reaction Dynamics of Triplet PyrimidinesYang, Chunfan ; Yu, Youqing ; Liu, Kunhui ; Song, Di ; Wu, Lidan ; Su, HongmeiThe journal of physical chemistry. A, Molecules, spectroscopy, kinetics, environment, & general theory, 2011-06, Vol.115 (21), p.5335-5345 [Periódico revisado por pares]United States: American Chemical SocietyTexto completo disponível |
9 |
Material Type: Artigo
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2-(2-Thienyl)-5,6-dihydroxy-4-carboxypyrimidines as Inhibitors of the Hepatitis C Virus NS5B Polymerase: Discovery, SAR, Modeling, and MutagenesisKoch, Uwe ; Attenni, Barbara ; Malancona, Savina ; Colarusso, Stefania ; Conte, Immacolata ; Di Filippo, Marcello ; Harper, Steven ; Pacini, Barbara ; Giomini, Claudia ; Thomas, Steven ; Incitti, Ilario ; Tomei, Licia ; De Francesco, Raffaele ; Altamura, Sergio ; Matassa, Victor G ; Narjes, FrankJournal of medicinal chemistry, 2006-03, Vol.49 (5), p.1693-1705 [Periódico revisado por pares]United States: American Chemical SocietyTexto completo disponível |
10 |
Material Type: Artigo
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2-(2,6-Dihalophenyl)-3-(pyrimidin-2-yl)-1,3-thiazolidin-4-ones as non-nucleoside HIV-1 reverse transcriptase inhibitorsRao, A ; Balzarini, J ; Carbone, A ; Chimirri, A ; De Clercq, E ; Monforte, A.M ; Monforte, P ; Pannecouque, C ; Zappalà, MAntiviral research, 2004-08, Vol.63 (2), p.79-84 [Periódico revisado por pares]Amsterdam: Elsevier B.VTexto completo disponível |