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Material Type: Artigo
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Modulation of endogenous opioid signaling by inhibitors of puromycin-sensitive aminopeptidaseSingh, Rohit ; Jiang, Rongrong ; Williams, Jessica ; Dobariya, Prakashkumar ; Hanak, Filip ; Xie, Jiashu ; Rothwell, Patrick E. ; Vince, Robert ; More, Swati S.European journal of medicinal chemistry, 2024-09, Vol.275, p.116604, Article 116604 [Periódico revisado por pares]Elsevier Masson SASTexto completo disponível |
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Material Type: Artigo
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Enhanced Sequence-Specific DNA Recognition Using Oligodeoxynucleotide-Benzimidazole ConjugatesSur, Souvik ; Pujari, Suresh ; Ranjan, Nihar ; Azankia Temgoua, Lidivine ; Wicks, Sarah L. ; Conner, Andrea ; Arya, Dev P.ACS bio & med chem au, 2024-06, Vol.4 (3), p.154-164 [Periódico revisado por pares]American Chemical SocietyTexto completo disponível |
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Material Type: Artigo
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Iodinated 4,4’‐Bipyridines with Antiproliferative Activity Against Melanoma Cell LinesPeluso, Paola ; Mamane, Victor ; Spissu, Ylenia ; Casu, Giuseppina ; Dessì, Alessandro ; Dallocchio, Roberto ; Sechi, Barbara ; Palmieri, Giuseppe ; Rozzo, CarlaChemMedChem, 2024-06, Vol.19 (12), p.e202300662-n/a [Periódico revisado por pares]Germany: Wiley Subscription Services, IncTexto completo disponível |
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Material Type: Artigo
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Spiro‐Acridine Compound as a Pteridine Reductase 1 Inhibitor: in silico Target Fishing and in vitro StudiesOliveira Viana, Jéssika ; Sena Mendes, Marina ; Santos Castilho, Marcelo ; Olímpio de Moura, Ricardo ; Guimarães Barbosa, EuzébioChemMedChem, 2024-06, Vol.19 (11), p.e202300545-n/a [Periódico revisado por pares]Germany: Wiley Subscription Services, IncTexto completo disponível |
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Material Type: Artigo
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Synthesis and antiproliferative evaluation of novel 3,5,8-trisubstituted coumarins against breast cancerSalem, Manar G ; Alqahtani, Alaa M ; Mali, Suraj N ; Alshwyeh, Hussah Abdullah ; Jawarkar, Rahul D ; Altamimi, Abdulmalik S ; Alshawwa, Samar Z ; Al-Olayan, Ebtesam ; Saied, Essa M ; Youssef, Mohamed FFuture medicinal chemistry, 2024-06, Vol.16 (11), p.1053-1073 [Periódico revisado por pares]England: Newlands Press LtdTexto completo disponível |
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Material Type: Artigo
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Synthesis and anti‐SARS‐CoV‐2 activity of amino acid modified cephalotaxine derivativesSi, Min ; An, Meidi ; Xia, Zhaomin ; Mo, Xiaoxue ; Lu, Jiayu ; He, Huaizhen ; Wang, ChengChemical biology & drug design, 2024-06, Vol.103 (6), p.e14566-n/a [Periódico revisado por pares]Texto completo disponível |
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Material Type: Artigo
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Tetrahydropyridine LIMK inhibitors: Structure activity studies and biological characterizationChampiré, Anthony ; Berabez, Rayan ; Braka, Abdennour ; Cosson, Aurélie ; Corret, Justine ; Girardin, Caroline ; Serrano, Amandine ; Aci-Sèche, Samia ; Bonnet, Pascal ; Josselin, Béatrice ; Brindeau, Pierre ; Ruchaud, Sandrine ; Leguevel, Rémy ; Chatterjee, Deep ; Mathea, Sebastian ; Knapp, Stefan ; Brion, Régis ; Verrecchia, Franck ; Vallée, Béatrice ; Plé, Karen ; Bénédetti, Hélène ; Routier, SylvainEuropean journal of medicinal chemistry, 2024-05, Vol.271, p.116391-116391, Article 116391 [Periódico revisado por pares]France: Elsevier Masson SASTexto completo disponível |
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Material Type: Artigo
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Anti-Aging Potential of the Two Major Flavonoids Occurring in Asian Water Lily Using In Vitro and In Silico Molecular Modeling AssessmentsNutho, Bodee ; Tungmunnithum, DuangjaiAntioxidants, 2024-05, Vol.13 (5), p.601 [Periódico revisado por pares]Switzerland: MDPI AGTexto completo disponível |
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Material Type: Artigo
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The Histone Deacetylase Family: Structural Features and Application of Combined Computational MethodsCurcio, Antonio ; Rocca, Roberta ; Alcaro, Stefano ; Artese, AnnaPharmaceuticals (Basel, Switzerland), 2024-05, Vol.17 (5), p.620 [Periódico revisado por pares]Switzerland: MDPI AGTexto completo disponível |
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Material Type: Artigo
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The emergence of machine learning force fields in drug designChen, Mingan ; Jiang, Xinyu ; Zhang, Lehan ; Chen, Xiaoxu ; Wen, Yiming ; Gu, Zhiyong ; Li, Xutong ; Zheng, MingyueMedicinal research reviews, 2024-05, Vol.44 (3), p.1147-1182 [Periódico revisado por pares]United States: Wiley Subscription Services, IncTexto completo disponível |