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1 |
Material Type: Artigo
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Further studies on analgesic activity of cyclic imidesFilho, Valdir Cechinel ; Corrêa, Rogério ; Vaz, Zulma ; Calixto, João Batista ; Nunes, Ricardo Jose ; Pinheiro, Tânia Rosely ; Andricopulo, Adriano Defini ; Yunes, Rosendo AugustoFarmaco (Società chimica italiana : 1989), 1998-01, Vol.53 (1), p.55-57 [Periódico revisado por pares]Lausanne: Elsevier SASTexto completo disponível |
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Material Type: Artigo
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Structure−Activity Relationships for a Class of Inhibitors of Purine Nucleoside PhosphorylaseFarutin, Victor ; Masterson, Lori ; Andricopulo, Adriano D ; Cheng, Jianming ; Riley, Brad ; Hakimi, Ryan ; Frazer, Jack W ; Cordes, Eugene HJournal of medicinal chemistry, 1999-07, Vol.42 (13), p.2422-2431 [Periódico revisado por pares]Washington, DC: American Chemical SocietyTexto completo disponível |
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Material Type: Artigo
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Structure-Activity Relationships for the Design of Small-Molecule InhibitorsAndricopulo, Adriano D ; Montanari, Carlos AMini reviews in medicinal chemistry, 2005-06, Vol.5 (6), p.585-593 [Periódico revisado por pares]Netherlands: Bentham Science Publishers LtdTexto completo disponível |
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Material Type: Artigo
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2D Quantitative structure–activity relationship studies on a series of cholesteryl ester transfer protein inhibitorsCastilho, Marcelo S. ; Guido, Rafael V.C. ; Andricopulo, Adriano D.Bioorganic & medicinal chemistry, 2007-09, Vol.15 (18), p.6242-6252 [Periódico revisado por pares]Oxford: Elsevier LtdTexto completo disponível |
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Material Type: Artigo
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Anacardic acid derivatives as inhibitors of glyceraldehyde-3-phosphate dehydrogenase from Trypanosoma cruziPereira, Junia M. ; Severino, Richele P. ; Vieira, Paulo C. ; Fernandes, João B. ; da Silva, M. Fátima G.F. ; Zottis, Aderson ; Andricopulo, Adriano D. ; Oliva, Glaucius ; Corrêa, Arlene G.Bioorganic & medicinal chemistry, 2008-10, Vol.16 (19), p.8889-8895 [Periódico revisado por pares]Amsterdam: Elsevier LtdTexto completo disponível |
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Material Type: Artigo
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Convergent synthesis and cruzain inhibitory activity of novel 2-( N′-benzylidenehydrazino)-4-trifluoromethyl-pyrimidinesZanatta, Nilo ; Amaral, Simone S. ; dos Santos, Josiane M. ; de Mello, Débora L. ; Fernandes, Liana da S. ; Bonacorso, Helio G. ; Martins, Marcos A.P. ; Andricopulo, Adriano D. ; Borchhardt, Deise M.Bioorganic & medicinal chemistry, 2008-12, Vol.16 (24), p.10236-10243 [Periódico revisado por pares]Amsterdam: Elsevier LtdTexto completo disponível |
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Material Type: Artigo
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Inhibition of Mycobacterium tuberculosis tyrosine phosphatase PtpA by synthetic chalcones: Kinetics, molecular modeling, toxicity and effect on growthMascarello, Alessandra ; Chiaradia, Louise Domeneghini ; Vernal, Javier ; Villarino, Andrea ; Guido, Rafael V.C. ; Perizzolo, Paulo ; Poirier, Valerie ; Wong, Dennis ; Martins, Priscila Graziela Alves ; Nunes, Ricardo José ; Yunes, Rosendo Augusto ; Andricopulo, Adriano Defini ; Av-Gay, Yossef ; Terenzi, HernánBioorganic & medicinal chemistry, 2010-06, Vol.18 (11), p.3783-3789 [Periódico revisado por pares]Amsterdam: Elsevier LtdTexto completo disponível |
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Material Type: Artigo
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Discovery of New Inhibitors of Schistosoma mansoni PNP by Pharmacophore-Based Virtual ScreeningPostigo, Matheus P ; Guido, Rafael V. C ; Oliva, Glaucius ; Castilho, Marcelo S ; da R. Pitta, Ivan ; de Albuquerque, Julianna F. C ; Andricopulo, Adriano DJournal of chemical information and modeling, 2010-09, Vol.50 (9), p.1693-1705 [Periódico revisado por pares]Washington, DC: American Chemical SocietyTexto completo disponível |
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Material Type: Artigo
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Acridone alkaloids as potent inhibitors of cathepsin VSeverino, Richele P. ; Guido, Rafael V.C. ; Marques, Emerson F. ; Brömme, Dieter ; da Silva, M. Fátima das G.F. ; Fernandes, João B. ; Andricopulo, Adriano D. ; Vieira, Paulo C.Bioorganic & medicinal chemistry, 2011-02, Vol.19 (4), p.1477-1481 [Periódico revisado por pares]Amsterdam: Elsevier LtdTexto completo disponível |
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Material Type: Artigo
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Synthesis, Biological Evaluation, And Molecular Modeling of Chalcone Derivatives As Potent Inhibitors of Mycobacterium tuberculosis Protein Tyrosine Phosphatases (PtpA and PtpB)Chiaradia, Louise Domeneghini ; Martins, Priscila Graziela Alves ; Cordeiro, Marlon Norberto Sechini ; Guido, Rafael Victorio Carvalho ; Ecco, Gabriela ; Andricopulo, Adriano Defini ; Yunes, Rosendo Augusto ; Vernal, Javier ; Nunes, Ricardo José ; Terenzi, HernánJournal of medicinal chemistry, 2012-01, Vol.55 (1), p.390-402 [Periódico revisado por pares]United States: American Chemical SocietyTexto completo disponível |