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1
[1, 8]-Naphthyridine derivatives as dual inhibitor of alkaline phosphatase and carbonic anhydrase
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Artigo
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[1, 8]-Naphthyridine derivatives as dual inhibitor of alkaline phosphatase and carbonic anhydrase

Alrokayan, Salman ; Hussain, Tajamul ; Alamery, Salman ; Mohammed, Arif Ahmed ; Mahmood, Abid ; Ejaz, Syeda Abida ; Langer, Peter ; Iqbal, Jamshed

BMC chemistry, 2023-10, Vol.17 (1), p.142-142, Article 142 [Periódico revisado por pares]

Cham: Springer International Publishing

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12 - Computer-aided methodologies to predict endocrine-disrupting potency of chemicals
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Capítulo de Livro
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12 - Computer-aided methodologies to predict endocrine-disrupting potency of chemicals

Roncaglioni, A. ; Benfenati, E.

Endocrine-disrupting chemicals in food, 2009, p.306-321

Elsevier Ltd

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3
1,2,4- and 1,3,4-Oxadiazoles as Scaffolds in the Development of Antiparasitic Agents
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1,2,4- and 1,3,4-Oxadiazoles as Scaffolds in the Development of Antiparasitic Agents

Pitasse-Santos, Paulo ; Sueth-Santiago, Vitor ; Lima, Marco

Journal of the Brazilian Chemical Society, 2018-03, Vol.29 (3), p.435-456 [Periódico revisado por pares]

Sociedade Brasileira de Química

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4
1,8‐Naphthalimide: A Potent DNA Intercalator and Target for Cancer Therapy
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1,8‐Naphthalimide: A Potent DNA Intercalator and Target for Cancer Therapy

Tandon, Runjhun ; Luxami, Vijay ; Kaur, Harsovin ; Tandon, Nitin ; Paul, Kamaldeep

Chemical record, 2017-10, Vol.17 (10), p.956-993 [Periódico revisado por pares]

United States: Wiley Subscription Services, Inc

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5
19-, an ent-abietane diterpene diepoxide, inhibits the growth of bladder cancer T24 cells through DNA damage
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Artigo
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19-, an ent-abietane diterpene diepoxide, inhibits the growth of bladder cancer T24 cells through DNA damage

Wang, Ke ; Yang, Juan-Cheng ; Jang, Yeong-Jiunn ; Chen, Guan-Yu ; Zhang, Ya-Jing ; Dai, Yun-Hao ; Zhang, Da-Yong ; Wu, Yang-Chang

PloS one, 2021-03, Vol.16 (3), p.e0248468 [Periódico revisado por pares]

Public Library of Science

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6
19-(Benzyloxy)-19-oxojolkinolide B (19-BJB), an ent-abietane diterpene diepoxide, inhibits the growth of bladder cancer T24 cells through DNA damage
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Artigo
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19-(Benzyloxy)-19-oxojolkinolide B (19-BJB), an ent-abietane diterpene diepoxide, inhibits the growth of bladder cancer T24 cells through DNA damage

Wang, Ke ; Yang, Juan-Cheng ; Jang, Yeong-Jiunn ; Chen, Guan-Yu ; Zhang, Ya-Jing ; Dai, Yun-Hao ; Zhang, Da-Yong ; Wu, Yang-Chang Lebedeva, Irina V.

PloS one, 2021-03, Vol.16 (3), p.e0248468-e0248468 [Periódico revisado por pares]

United States: Public Library of Science

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7
1H chemical shift differences of Prelog-Djerassi lactone derivatives: DFT and NMR conformational studiesElectronic supplementary information (ESI) available. See DOI: 10.1039/c4ob02446j
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1H chemical shift differences of Prelog-Djerassi lactone derivatives: DFT and NMR conformational studiesElectronic supplementary information (ESI) available. See DOI: 10.1039/c4ob02446j

Aímola, Túlio J ; Lima, Dimas J. P ; Dias, Luiz C ; Tormena, Cláudio F ; Ferreira, Marco A. B

2015-02

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8
2-(2-Methylfuran-3-carboxamido)-3-phenylpropanoic acid, a potential CYP26A1 inhibitor to enhance all-trans retinoic acid-induced leukemia cell differentiation based on virtual screening and biological evaluation
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2-(2-Methylfuran-3-carboxamido)-3-phenylpropanoic acid, a potential CYP26A1 inhibitor to enhance all-trans retinoic acid-induced leukemia cell differentiation based on virtual screening and biological evaluation

Li, Fengrong ; Zhao, Dongmei ; Ren, Jinhong ; Hao, Feiyue ; Liu, Guyue ; Jin, Shengfei ; Jing, Yongkui ; Cheng, Maosheng

Bioorganic & medicinal chemistry, 2013-06, Vol.21 (11), p.3256-3261 [Periódico revisado por pares]

England: Elsevier Ltd

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9
2-aminobenzimidazoles for leishmaniasis: From initial hit discovery to in vivo profiling
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Artigo
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2-aminobenzimidazoles for leishmaniasis: From initial hit discovery to in vivo profiling

Ferreira, Rafael Augusto Alves ; Junior, Celso de Oliveira Rezende ; Martinez, Pablo David Grigol ; Koovits, Paul John ; Soares, Bruna Miranda ; Ferreira, Leonardo L G ; Michelan-Duarte, Simone ; Chelucci, Rafael Consolin ; Andricopulo, Adriano D ; Galuppo, Mariana K ; Uliana, Silvia R B ; Matheeussen, An ; Caljon, Guy ; Maes, Louis ; Campbell, Simon ; Kratz, Jadel M ; Mowbray, Charles E ; Dias, Luiz Carlos Croft, Simon L.

PLoS neglected tropical diseases, 2021-02, Vol.15 (2), p.e0009196 [Periódico revisado por pares]

United States: Public Library of Science

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10
2-octadecynoic acid as a dual life stage inhibitor of plasmodium infections and plasmodial fas-ii enzymes
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Artigo
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2-octadecynoic acid as a dual life stage inhibitor of plasmodium infections and plasmodial fas-ii enzymes

Carballeira, Néstor M ; Bwalya, Angela Gono ; Itoe, Maurice Ayamba ; Andricopulo, Adriano D ; Cordero-Maldonado, María Lorena ; Kaiser, Marcel ; Mota, Maria M ; Crawford, Alexander D ; Guido, Rafael V.C ; Tasdemir, Deniz

Bioorganic & Medicinal Chemistry Letters, 2014-09 [Periódico revisado por pares]

Elsevier BV

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