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1 |
Material Type: Artigo
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AI is a viable alternative to high throughput screening: a 318-target studyBernard, Denzil ; Morrison, Adrian ; Ng, Ho Leung ; Ahmed, Mostafa ; Anthis, Nicholas J. ; PrasadPrasad, Srimukh Veccham Krishna ; Shek, Stefani ; Lee, Andreia H. ; DeHaan, Nicholas ; Abramyan, Tigran M. ; Ghosh, Agnidipta ; Statsyuk, Alexander V. ; Caflisch, Amedeo ; Matheeussen, An ; Battistoni, Andrea ; Chini, Andrea ; Ilari, Andrea ; Foote, Andrea Talbot ; Samantha, Ariela ; ElSheikh, Assmaa ; Edelman, Benjamin L. ; Morten, Brianna C. ; Lempicki, Camille ; Chapman, Carly J. ; Partch, Carrie L. ; Huang, Chang ; Hu, Di ; Ortiz, Diana ; Dirksen, Dorian ; Lama, Eleonora ; Christensen, Emily M. ; Trakhtenberg, Ephraim F. ; Kroon, Erna Geessien ; Yu, Fang ; van den Akker, Focco ; Vizeacoumar, Franco J. ; Vizeacoumar, Frederick S. ; Mayer, Gaétan ; Girolimetti, Giulia ; Dahal, Gopal ; Bowman, Gregory R. ; Akk, Gustav ; Jafar-Nejad, Hamed ; Jung, Hoyoung ; Fan, Hua-Ying ; Arozarena, Imanol ; Ferreira, Jacob ; Siqueira-Neto, Jair L. ; Evans, Jay D. ; Wang, Jianghai ; So, Jonathan ; Gruber, Joshua J. ; Lasarte, Juan José ; Lescar, Julien ; Bogomolovas, Julijus ; Sistla, Jyothi C. ; Hopkins, Kevin M. ; Mostert, Konrad J. ; Rohde, Kyle H. ; Pusztai, Lajos ; Cowen, Leah E. ; Su, Leila ; Wert-Lamas, Leon ; Puchades-Carrasco, Leonor ; Zhuo, Ling ; Valli, Marilia ; Tye, Mark A. ; Wilson, Mark A. ; Alteen, Matthew G. ; Rizzi, Menico ; Paige, Mikell ; Matovic, Nick ; Horstmann, Nicola ; Khalaf, Noureddine Ben ; Sobrado, Pablo ; Chuong, Patrick ; Wu, Pengpeng ; Agogo-Mawuli, Percy ; Toogood, Peter ; von Hundelshausen, Philipp ; Lee, Pil H. ; Balaña-Fouce, Rafael ; Singh, Rakesh K. ; Tiwari, Rakesh Kumar ; Austin, Richard C. ; Bradley, Robert K. ; Reguera, Rosa Maria ; Uribe, Ruben Vazquez ; Gorgoglione, Ruggiero ; Geden, Sandra E. ; Chauhan, Shefali ; Shyng, Show-Ling ; Xu, Sophia Q. ; Gustincich, Stefano ; Marx, Steven O. ; Banerji, Versha ; Robinson, Victoria L. ; Gunasekharan, Vignesh ; Van Hung Le, Vuong ; Wu, XiaoyangScientific reports, 2024-04, Vol.14 (1), p.7526-16, Article 7526 [Periódico revisado por pares]England: Nature Publishing GroupTexto completo disponível |
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Material Type: Artigo
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Treatments for dengue: a Global Dengue Alliance to address unmet needsAnasir, Mohd Ishtiaq ; Angkasekwinai, Nasikarn ; Auewarakul, Prasert ; Avirutnan, Panisadee ; Bilbe, Graeme ; Charvillon, Fabienne Burgat ; Costa, Vivian Vasconcelos ; Croda, Julio ; Daher, Andre ; Das, Supratik ; Ellan, E.Kavithambigai ; Gani, Yasmin ; Garg, Pramod ; Uppal, Geetanjali ; Guruge, Dinuka ; Kalyanasundram, Jeevanathan ; Kratz, Jadel Müller ; Krieger, Marco A. ; Lapphra, Keswadee ; Lim, Steven Chee Loon ; Lodha, Rakesh ; Mahajan, Dinesh ; Malavige, Gathsaurie Neelika ; Mairiang, Dumrong ; Marques, Ernesto Torres D Azevedo ; Md Jelas, Nur Hana ; Medigeshi, Guruprasad R. ; Mohd Abd Razak, Mohd Ridzuan ; Mohd Zain, Rozainanee ; Mowbray, Charles ; Nischal, Neeraj ; Nogueira, Mauricio L. ; Noisakran, Sansanee ; Punyadee, Nuntaya ; Pedrique, Belen ; Piedagnel, Jean-Michel ; Punnawit Phongpitchanont, Surat ; Ramanaidu, Tilakbabu ; Ribeiro, Isabela ; Rose, Winsley ; Rupali, Priscilla ; Samal, Sweety ; Singh, Kavita ; Siqueira, Andre M. ; Sjö, Peter ; Sosa-Estani, Sergio ; Souza, Thiago Moreno L. ; Suppiah, Jeyanthi ; Syed Mohamed, Ami Fazlin ; Mohd Tahir, Nur Zaidah ; Tan, Terence Yew Chin ; Teixeira, Mauro M. ; Thayan, Ravindran ; Wadhwa, Nitya ; Wijewickrama, Ananda ; Mohamed Yusoff, Fazlina ; Zainol, MurizalThe Lancet global health, 2023-11, Vol.11 (11), p.e1680-e1681 [Periódico revisado por pares]Elsevier LtdTexto completo disponível |
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Material Type: Artigo
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Hit-to-lead optimization of a 2-aminobenzimidazole series as new candidates for chagas diseaseCelso de Oliveira Rezende Junior Pablo David Grigol Martinez; Rafael Augusto Alves Ferreira; Paul John Koovits; Bruna Miranda Soares; Leonardo Luiz Gomes Ferreira; Simone Michelan Duarte; Rafael Consolin Chelucci; Adriano Defini Andricopulo; An Matheeussen; Natascha Van Pelt; Guy Caljon; Louis Maes; Simon Campbell; Jadel Muller Kratz; Charles E Mowbray; Luiz Carlos DiasEuropean Journal of Medicinal Chemistry Issy-les-Moulineaux v. 246, p. 114925-1-114925-10 + supplementary data, Jan. 2023Issy-les-Moulineaux 2023Localização: IFSC - Inst. Física de São Carlos (PROD033848 )(Acessar) |
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Material Type: Artigo
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Effects of Lipophilicity and Structural Features on the Antiherpes Activity of Digitalis Cardenolides and DerivativesPádua, Rodrigo Maia ; Kratz, Jadel Müller ; Munkert, Jennifer ; Bertol, Jéssica Wildgrube ; Rigotto, Caroline ; Schuster, Daniela ; Maltarollo, Vinícius Gonçalves ; Kreis, Wolfgang ; Simões, Cláudia Maria Oliveira ; Braga, Fernão CastroChemistry & biodiversity, 2022-10, Vol.19 (10), p.e202200411-n/a [Periódico revisado por pares]Weinheim: Wiley Subscription Services, IncTexto completo disponível |
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Material Type: Dataset
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In vitro intestinal permeability studies, pharmacokinetics and tissue distribution of 6-methylcoumarin after oral and intraperitoneal administration in Wistar ratsCárdenas, Paola Andrea ; Kratz, Jadel Müller ; Hernández, Aura ; Costa, Geison Modesti ; Ospina, Luis Fernando ; Baena, Yolima ; Simões, Cláudia Maria Oliveira ; Jimenez-Kairuz, Álvaro ; Aragon, MarcelaSciELO journals 2022Texto completo disponível |
6 |
Material Type: Artigo de Congresso
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Indoles hit-to-lead for chagas disease lessons learned within the LOLA consortiumLuiza Cruz Adriana Corrêa da Silva; Clarissa Feltrin; Maria Dichiara; Lori Ferrins; Carolina Borsoi Moraes; Peter Sjo; Adriano Defini Andricopulo; Charles Mowbray; Ramon Guerra de Oliveira; Marco Aurélio Dessoy; Deborah Araújo dos Santos; Luiz Fernando Nascimento de Oliveira; María Cruz Mollo; Eun Lee; Simone Michelan Duarte; Renata Krogh Andricopulo; Rafael Consolin Chelucci; Leonardo Luiz Gomes Ferreira; Jadel Muller Kratz; Luiz Carlos Dias; Brazilian Symposium on Medicinal Chemistry - BrazMedChem (10. 2022 Campinas)Anais eletrônicos Campinas : Galoá, 2022Campinas Galoá 2022Acesso online. A biblioteca também possui exemplares impressos. |
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Material Type: Artigo
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Drug discovery for chagas disease: A viewpointKratz, Jadel MüllerActa tropica, 2019-10, Vol.198, p.105107-105107, Article 105107 [Periódico revisado por pares]Netherlands: Elsevier B.VTexto completo disponível |
8 |
Material Type: Artigo
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Clinical and pharmacological profile of benznidazole for treatment of Chagas diseaseMüller Kratz, Jadel ; Garcia Bournissen, Facundo ; Forsyth, Colin J. ; Sosa-Estani, SergioExpert review of clinical pharmacology, 2018-10, Vol.11 (10), p.943-957 [Periódico revisado por pares]England: Taylor & FrancisSem texto completo |
9 |
Material Type: Artigo
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Pharmacokinetics of Saquinavir Mesylate from Oral Self-Emulsifying Lipid-Based Delivery SystemsCaon, Thiago ; Kratz, Jadel Muller ; Kuminek, Gislaine ; Heller, Melina ; Micke, Gustavo Amadeu ; de Araujo, Bibiana Verlindo ; Koester, Letícia Scherer ; Simões, Cláudia Maria OliveiraEuropean journal of drug metabolism and pharmacokinetics, 2017-02, Vol.42 (1), p.135-141 [Periódico revisado por pares]Cham: Springer International PublishingTexto completo disponível |
10 |
Material Type: Artigo
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In vitro intestinal permeability studies, pharmacokinetics and tissue distribution of 6-methylcoumarin after oral and intraperitoneal administration in Wistar ratsCárdenas, Paola Andrea ; Kratz, Jadel Müller ; Hernández, Aura ; Costa, Geison Modesti ; Ospina, Luis Fernando ; Baena, Yolima ; Simões, Cláudia Maria Oliveira ; Jimenez-Kairuz, Álvaro ; Aragon, MarcelaBrazilian Journal of Pharmaceutical Sciences, 2017-01, Vol.53 (1) [Periódico revisado por pares]Sao Paulo: Universidade de Sao Paulo Faculdade de CienciasTexto completo disponível |