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1
1-[5-(2-Fluorophenyl)-1-(pyridin-3-ylsulfonyl)-1H-pyrrol-3-yl]-N-methylmethanamine monofumarate (TAK-438), a novel and potent potassium-competitive acid blocker for the treatment of acid-related diseases
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Artigo
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1-[5-(2-Fluorophenyl)-1-(pyridin-3-ylsulfonyl)-1H-pyrrol-3-yl]-N-methylmethanamine monofumarate (TAK-438), a novel and potent potassium-competitive acid blocker for the treatment of acid-related diseases

Hori, Yasunobu ; Imanishi, Akio ; Matsukawa, Jun ; Tsukimi, Yasuhiro ; Nishida, Haruyuki ; Arikawa, Yasuyoshi ; Hirase, Keizo ; Kajino, Masahiro ; Inatomi, Nobuhiro

The Journal of pharmacology and experimental therapeutics, 2010-10, Vol.335 (1), p.231-238 [Periódico revisado por pares]

United States

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2
1, 5-Benzoxathiepin Derivatives. II. Synthesis and Serotonin S2-Receptor-Blocking Activity of Aminoalkyl-Substituted 3, 4-Dihydro-2H-1, 5-benzoxathiepin-3-ols and Related Compounds
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Artigo
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1, 5-Benzoxathiepin Derivatives. II. Synthesis and Serotonin S2-Receptor-Blocking Activity of Aminoalkyl-Substituted 3, 4-Dihydro-2H-1, 5-benzoxathiepin-3-ols and Related Compounds

SUGIHARA, HIROSADA ; MABUCHI, HIROSHI ; HIRATA, MINORU ; IMAMOTO, TETSUJI ; KAWAMATSU, YUTAKA

Chemical and Pharmaceutical Bulletin, 1987/05/25, Vol.35(5), pp.1930-1952 [Periódico revisado por pares]

Tokyo: The Pharmaceutical Society of Japan

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3
1, 5-Benzoxathiepin Derivatives. III. Optical Resolution of Methyl (±)-cis-3-Hydroxy-4-[3-(4-phenyl-1-piperazinyl)propyl]-3, 4-dihydro-2H-1, 5-benzoxathiepin-4-carboxylate Hydrochloride ((±)-CV-5197) with Selective 5-Hydroxytryptamine2(5-HT2)-Antagonistic Activity
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Artigo
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1, 5-Benzoxathiepin Derivatives. III. Optical Resolution of Methyl (±)-cis-3-Hydroxy-4-[3-(4-phenyl-1-piperazinyl)propyl]-3, 4-dihydro-2H-1, 5-benzoxathiepin-4-carboxylate Hydrochloride ((±)-CV-5197) with Selective 5-Hydroxytryptamine2(5-HT2)-Antagonistic Activity

KORI, Masakuni ; KAMIYA, Kazuhide ; KURIHARA, Etsuo ; SUGIHARA, Hirosada

Chemical and Pharmaceutical Bulletin, 1991/04/25, Vol.39(4), pp.922-926 [Periódico revisado por pares]

Tokyo: The Pharmaceutical Society of Japan

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4
1-(5-Carboxyindazol-1-yl)propan-2-ones as dual inhibitors of cytosolic phospholipase A 2 α and fatty acid amide hydrolase: bioisosteric replacement of the carboxylic acid moiety
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1-(5-Carboxyindazol-1-yl)propan-2-ones as dual inhibitors of cytosolic phospholipase A 2 α and fatty acid amide hydrolase: bioisosteric replacement of the carboxylic acid moiety

Althaus, Jan ; Hake, Theresa ; Hanekamp, Walburga ; Lehr, Matthias

Journal of enzyme inhibition and medicinal chemistry, 2016-11, Vol.31 (sup1), p.131-140 [Periódico revisado por pares]

England

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5
1,102 pounds
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magazinearticle
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1,102 pounds

The New York times upfront, 2020-02, Vol.152 (9), p.4

Scholastic, Inc

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6
1,1′-Disubstituted Ferrocenes as Molecular Hinges in Mono- and Bivalent Dopamine Receptor Ligands
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1,1′-Disubstituted Ferrocenes as Molecular Hinges in Mono- and Bivalent Dopamine Receptor Ligands

Huber, Daniela ; Hübner, Harald ; Gmeiner, Peter

Journal of medicinal chemistry, 2009-11, Vol.52 (21), p.6860-6870 [Periódico revisado por pares]

United States: American Chemical Society

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7
1,2,3- dl-Tricarboxycyclopentene-1 and other inhibitors of cis-aconitase
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1,2,3- dl-Tricarboxycyclopentene-1 and other inhibitors of cis-aconitase

Gawron, Oscar ; Birckbichler, Paul J.

Archives of biochemistry and biophysics, 1971-12, Vol.147 (2), p.772-780 [Periódico revisado por pares]

United States: Elsevier Inc

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8
1,25-dihydroxyvitamin D radioreceptor assay using bovine mammary gland receptor and non-high performance liquid chromatographic purification
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Artigo
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1,25-dihydroxyvitamin D radioreceptor assay using bovine mammary gland receptor and non-high performance liquid chromatographic purification

WATANABE, Y ; KUBOTA, T ; SUZUMURA, E ; SUZUKI, T ; YONEZAWA, M ; ISHIGAMI, T ; ICHIKAWA, M ; SEINO, Y

Clinica chimica acta, 1994-03, Vol.225 (2), p.187-194 [Periódico revisado por pares]

Shannon: Elsevier

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9
1,25-Dihydroxyvitamin D3 induces 25-hydroxyvitamin D3-24-hydroxylase in a cultured monkey kidney cell line (LLC-MK2) apparently deficient in the high affinity receptor for the hormone
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Artigo
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1,25-Dihydroxyvitamin D3 induces 25-hydroxyvitamin D3-24-hydroxylase in a cultured monkey kidney cell line (LLC-MK2) apparently deficient in the high affinity receptor for the hormone

Chandler, J S ; Chandler, S K ; Pike, J W ; Haussler, M R

The Journal of biological chemistry, 1984-02, Vol.259 (4), p.2214-2222 [Periódico revisado por pares]

Bethesda, MD: Elsevier Inc

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10
1,25-Dihydroxyvitamin D3 Negatively Regulates the Inflammatory Response to Porcine Epidemic Diarrhea Virus Infection by Inhibiting NF-κB and JAK/STAT Signaling Pathway in IPEC-J2 Porcine Epithelial Cells
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1,25-Dihydroxyvitamin D3 Negatively Regulates the Inflammatory Response to Porcine Epidemic Diarrhea Virus Infection by Inhibiting NF-κB and JAK/STAT Signaling Pathway in IPEC-J2 Porcine Epithelial Cells

Yang, Jiwen ; Chen, Daiwen ; Tian, Gang ; Mao, Xiangbing ; He, Jun ; Zheng, Ping ; Yu, Jie ; Luo, Yuheng ; Luo, Junqiu ; Huang, Zhiqing ; Wu, Aimin ; Yan, Hui ; Yu, Bing

International journal of molecular sciences, 2022-09, Vol.23 (18), p.10603 [Periódico revisado por pares]

Basel: MDPI AG

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Deste Autor:

  1. Moreno, A
  2. Garbossa, C
  3. Andrade, A
  4. Moretti, A
  5. Martins, S

Buscando em bases de dados remotas. Favor aguardar.